PRKAA1/AMPKα1-driven glycolysis in endothelial cells exposed to disturbed flow protects against atherosclerosis

Nat Commun. 2018 Nov 7;9(1):4667. doi: 10.1038/s41467-018-07132-x.

Abstract

Increased aerobic glycolysis in endothelial cells of atheroprone areas of blood vessels has been hypothesized to drive increased inflammation and lesion burden but direct links remain to be established. Here we show that endothelial cells exposed to disturbed flow in vivo and in vitro exhibit increased levels of protein kinase AMP-activated (PRKA)/AMP-activated protein kinases (AMPKs). Selective deletion of endothelial Prkaa1, coding for protein kinase AMP-activated catalytic subunit alpha1, reduces glycolysis, compromises endothelial cell proliferation, and accelerates the formation of atherosclerotic lesions in hyperlipidemic mice. Rescue of the impaired glycolysis in Prkaa1-deficient endothelial cells through Slc2a1 overexpression enhances endothelial cell viability and integrity of the endothelial cell barrier, and reverses susceptibility to atherosclerosis. In human endothelial cells, PRKAA1 is upregulated by disturbed flow, and silencing PRKAA1 reduces glycolysis and endothelial viability. Collectively, these results suggest that increased glycolysis in the endothelium of atheroprone arteries is a protective mechanism.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • AMP-Activated Protein Kinases / metabolism*
  • Animals
  • Apolipoproteins E / deficiency
  • Apolipoproteins E / metabolism
  • Atherosclerosis / enzymology*
  • Atherosclerosis / prevention & control*
  • Endothelial Cells / enzymology*
  • Endothelial Cells / metabolism
  • Endothelial Cells / pathology
  • Glucose Transporter Type 1 / metabolism
  • Glycolysis*
  • Human Umbilical Vein Endothelial Cells / metabolism
  • Humans
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Models, Biological
  • Rheology*

Substances

  • Apolipoproteins E
  • Glucose Transporter Type 1
  • Slc2a1 protein, mouse
  • AMPK alpha1 subunit, mouse
  • AMP-Activated Protein Kinases
  • PRKAA1 protein, human