RORα suppresses interleukin-6-mediated hepatic acute phase response

Sci Rep. 2019 Aug 13;9(1):11798. doi: 10.1038/s41598-019-48171-8.

Abstract

Acute liver failure (ALF) is characterized by loss of liver function in response to sustained augmentation of the acute-phase response (APR) in the liver, which can progress even to death. Although the inflammatory interleukin-6 (IL-6)-axis is a crucial factor that drives the hepatic APR by releasing diverse acute-phase proteins (APPs), therapeutic strategies to block the IL-6-STAT3-mediated APR are not well developed. Here, we show that the nuclear receptor retinoic acid-related orphan receptor α (RORα) limits APR-mediated liver injury by inhibiting the hepatic IL-6-STAT3 signaling pathway. Administration of JC1-40, an RORα activator, diminished diethylnitrosamine-induced acute liver injury and repressed transcriptional expression of APPs such as CXCL1 and LCN2 in mice. IL-6-mediated activation of STAT3 was repressed after RORα activation by either adenoviral infusion of RORα or JC1-40 treatment in primary hepatocytes. Activation of RORα decreased transcriptional expression of IL-6 receptor α, an upstream activator of STAT3, both in vitro and in vivo. This may be one mechanism underlying the RORα-mediated inhibition of STAT3. Taken together, our results suggest that RORα is a regulator of the hepatic IL-6-STAT3 signaling pathway and may be a new therapeutic target for treating APR-associated inflammatory ALF.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acute-Phase Reaction / genetics
  • Adenoviridae / genetics
  • Animals
  • Chemical and Drug Induced Liver Injury / drug therapy*
  • Chemical and Drug Induced Liver Injury / genetics
  • Chemical and Drug Induced Liver Injury / pathology
  • Chemokine CXCL1 / genetics
  • Deoxyuracil Nucleotides / pharmacology
  • Diethylnitrosamine / toxicity
  • Disease Models, Animal
  • Gene Expression Regulation / drug effects
  • Hepatocytes / drug effects
  • Humans
  • Hydroxycholesterols / pharmacology
  • Interleukin-6 / genetics*
  • Liver / injuries
  • Liver / metabolism
  • Liver / pathology
  • Liver Failure, Acute / drug therapy*
  • Liver Failure, Acute / genetics
  • Liver Failure, Acute / pathology
  • Mice
  • Nuclear Receptor Subfamily 1, Group F, Member 1 / antagonists & inhibitors
  • Nuclear Receptor Subfamily 1, Group F, Member 1 / genetics*
  • Primary Cell Culture
  • STAT3 Transcription Factor / genetics*
  • Signal Transduction / drug effects

Substances

  • Chemokine CXCL1
  • Cxcl1 protein, mouse
  • Deoxyuracil Nucleotides
  • Hydroxycholesterols
  • Interleukin-6
  • Nuclear Receptor Subfamily 1, Group F, Member 1
  • Rora protein, mouse
  • STAT3 Transcription Factor
  • JC 40
  • Diethylnitrosamine