Protective effects of Platycodon grandiflorus polysaccharides against apoptosis induced by carbonyl cyanide 3-chlorophenylhydrazone in 3D4/21 cells

Int J Biol Macromol. 2019 Dec 1:141:1220-1227. doi: 10.1016/j.ijbiomac.2019.09.086. Epub 2019 Sep 12.

Abstract

This study aimed to investigate the potential protective effects of Platycodon grandiflorus polysaccharide (PGPS) on carbonyl cyanide 3-chlorophenylhydrazone (CCCP)-induced mitochondrial apoptosis in 3D4/21 cells. Apoptosis-related indicators such as cell viability, apoptosis rate, mitochondrial membrane potential (MMP), and apoptosis-related protein were examined. Results indicated that PGPSt can inhibit CCCP-induced cell damage, with cell-survival rate reaching 81% and apoptotic rate decreasing to 23%. Nuclear deformation was also significantly reduced in the PGPSt group, and changes in MMP were inhibited by PGPSt. Further analyses showed that the protein expression of Caspase-9 and Bcl-2 increased and the expression of cleaved Caspase-3 decreased, indicating that PGPSt significantly inhibited the CCCP-induced change in apoptotic protein expression. All these results suggested that PGPSt can antagonize 3D4/21 cell apoptosis by restoring MMP, protecting the integrity of nuclear morphology, and increasing Bcl-2 expression.

Keywords: 3D4/21 cells; Mitochondrial apoptosis pathway; Platycodon grandiflorus polysaccharides.

MeSH terms

  • Apoptosis / drug effects*
  • Caspase 3 / metabolism
  • Caspase 9 / metabolism
  • Cell Line
  • Cell Proliferation / drug effects
  • Cytoprotection / drug effects*
  • Gene Expression Regulation, Enzymologic / drug effects
  • Hydrazones / toxicity*
  • Membrane Potential, Mitochondrial / drug effects
  • Platycodon / chemistry*
  • Polysaccharides / pharmacology*
  • Proto-Oncogene Proteins c-bcl-2 / metabolism

Substances

  • Hydrazones
  • Polysaccharides
  • Proto-Oncogene Proteins c-bcl-2
  • carbonyl 3-chlorophenylhydrazone
  • Caspase 3
  • Caspase 9