Microenvironment-Responsive Small-Molecule Probe for Pulmonary Fibrosis Detection

Anal Chem. 2020 Jan 7;92(1):699-706. doi: 10.1021/acs.analchem.9b02264. Epub 2019 Dec 13.

Abstract

Pulmonary fibrosis (PF) is a fatal disease with increasing prevalence. Nonradioactive and noninvasive diagnosis of PF at an early stage can improve the prognosis but represents a daunting challenge. Up-regulation of nitric oxide (NO) is a typical microenvironmental feature of PF. Here, we report a small-molecule probe, PNO1, that can fluorogenically sense this microenvironmental feature for PF diagnosis. We demonstrate that PNO1 fluorescence is 6-fold higher in PF-diseased mice lungs than in normal-control groups. In addition to this in vivo result, PNO1 can also be applied in vitro to detect PF-diseased cells and ex vivo to detect PF-diseased tissues from clinical patients. These results highlight PNO1 as a complement to the traditional immunostaining-based methods for PF detection to facilitate quick screening for anti-PF drug candidates.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line
  • Fluorescent Dyes / administration & dosage
  • Fluorescent Dyes / chemical synthesis
  • Fluorescent Dyes / chemistry*
  • Injections, Intravenous
  • Mice
  • Molecular Structure
  • Nitric Oxide / analysis
  • Nitric Oxide / metabolism
  • Optical Imaging
  • Pulmonary Fibrosis / diagnosis*
  • Pulmonary Fibrosis / metabolism
  • Small Molecule Libraries / administration & dosage
  • Small Molecule Libraries / chemical synthesis
  • Small Molecule Libraries / chemistry*

Substances

  • Fluorescent Dyes
  • Small Molecule Libraries
  • Nitric Oxide