Rosmarinic Acid/ Blue Light Combination Treatment Inhibits Head and Neck Squamous Cell Carcinoma In Vitro

Anticancer Res. 2020 Feb;40(2):751-758. doi: 10.21873/anticanres.14006.

Abstract

Background/aim: This study investigated a novel combined therapy of rosmarinic acid (RA)/blue light on head and neck squamous cell carcinoma (HNSCC) cell proliferation in vitro.

Materials and methods: HNSCC cells were exposed to BL (500 mW/cm2) for 90 s, and incubated with 80 μg/ml RA for 1 hour. Cell viability was determined after 24 h using WST-1 assay. Western blot was used to detect treatment-induced changes in epidermal growth factor receptor (EGFR) activation. Hydrogen peroxide (H2O2) and nitric oxide levels were quantified using CM-H2DCFH-DA assays. Apoptosis was assessed using Annexin V/PI staining and flow cytometry.

Results: RA/blue light treatment resulted in a significant reduction in cell viability, EGFR activation and H2O2 levels in all HNSCC cell lines. However, no significant changes in NO production or apoptosis induction were found.

Conclusion: RA/blue light effectively decreased HNSCC cell proliferation through reduction in EGFR activation and H2O2 production, and not via induction of apoptosis.

Keywords: EGF receptor; Head and neck cancer; light; oxidative stress; phytochemicals.

MeSH terms

  • Cell Line, Tumor
  • Cell Proliferation / drug effects
  • Cinnamates / pharmacology*
  • Combined Modality Therapy
  • Depsides / pharmacology*
  • Enzyme Activation / drug effects
  • ErbB Receptors / metabolism
  • Head and Neck Neoplasms / drug therapy
  • Head and Neck Neoplasms / pathology
  • Head and Neck Neoplasms / therapy*
  • Humans
  • Nitric Oxide / metabolism
  • Oxidative Stress / drug effects
  • Phototherapy / methods*
  • Rosmarinic Acid
  • Squamous Cell Carcinoma of Head and Neck / drug therapy
  • Squamous Cell Carcinoma of Head and Neck / pathology
  • Squamous Cell Carcinoma of Head and Neck / therapy*

Substances

  • Cinnamates
  • Depsides
  • Nitric Oxide
  • EGFR protein, human
  • ErbB Receptors