Triamcinolone acetonide loaded-cationic nano-lipoidal formulation for uveitis: Evidences of improved biopharmaceutical performance and anti-inflammatory activity

Colloids Surf B Biointerfaces. 2020 Jun:190:110902. doi: 10.1016/j.colsurfb.2020.110902. Epub 2020 Feb 25.

Abstract

Topical administration of corticosteroids is the cornerstone treatment of anterior uveitis, but poor corneal penetration and retention cause hindrance in their therapeutic utility. The conventional eye drops are less valuable in conditions where inflammation reaches deeper regions of the eye. Therefore, there is a clear need for an effective drug delivery system, which can increase corticosteroid penetration after topical application. To address this, cationic nanostructured lipid carriers of the drug triamcinolone acetonide (cTA-NLC) were prepared. The cTA-NLC were prepared by a hot microemulsion method and evaluated for drug release, permeation, cell uptake, cytotoxicity, anti-inflammatory activity and ocular irritancy. The cTA-NLC are nanometric in size (< 200 nm), with a zeta potential of about +35 mv and % drug EE of 88 %. The nanocarriers exhibited slow and sustained release of around 84 % in 24 h and transcorneal drug permeation of 51 % in 8 h. The nanocarriers exhibited no cytotoxicity (% cell viability of>90 %). The cell uptake study showed that nanocarriers could retain inside the cells for 24 h. The developed formulation could significantly reduce the TNF-α level in LPS induced inflamed cells. The studies indicated that cTA-NLC could be a promising option for the topical treatment of uveitis.

Keywords: Corneal permeation; Human corneal fibroblast cells (HCF); Nanostructured lipid nanocarriers; Triamcinolone acetonide; Uveitis.

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / chemistry
  • Anti-Inflammatory Agents / pharmacology*
  • Biological Products / chemistry
  • Biological Products / pharmacology*
  • Cations / chemistry
  • Cell Survival / drug effects
  • Cells, Cultured
  • Chickens
  • Dose-Response Relationship, Drug
  • Drug Liberation
  • Humans
  • Lipids / chemistry*
  • Nanoparticles / chemistry*
  • Particle Size
  • Structure-Activity Relationship
  • Surface Properties
  • Triamcinolone Acetonide / chemistry
  • Triamcinolone Acetonide / pharmacology*
  • Tumor Necrosis Factor-alpha / antagonists & inhibitors
  • Uveitis / drug therapy*
  • Uveitis / pathology

Substances

  • Anti-Inflammatory Agents
  • Biological Products
  • Cations
  • Lipids
  • Tumor Necrosis Factor-alpha
  • Triamcinolone Acetonide