Nintedanib-induced glomerular microangiopathy: a case report

CEN Case Rep. 2020 Nov;9(4):295-300. doi: 10.1007/s13730-020-00474-w. Epub 2020 Apr 11.

Abstract

Nintedanib, a triple tyrosine kinase inhibitor of vascular endothelial growth factor receptor, platelet-derived growth factor receptor, and fibroblast growth factor receptor, has been used in idiopathic pulmonary fibrosis and adenocarcinoma in advanced non-small cell lung cancer. Although vascular endothelial growth factor inhibitors have been reported to cause endothelial injury and glomerular microangiopathy, nintedanib-induced glomerular microangiopathy has not been reported. A 68-year-old man with a history of primary aldosteronism, idiopathic pulmonary fibrosis, and pleomorphic carcinoma of the lung developed proteinuria and leg edema after nintedanib initiation. Kidney biopsy revealed prominent endothelial and mesangial injury. Proteinuria improved after nintedanib withdrawal. To the best of our knowledge, this is the second case report of nintedanib-induced glomerular microangiopathy. Although the incidence of nephropathy among patients receiving nintedanib is unknown at this moment, we recommend monitoring urinary protein excretion and blood pressure in patients receiving nintedanib and performing kidney biopsy to determine any histopathological change.

Keywords: Glomerular microangiopathy; Nintedanib; Onconephrology; Proteinuria; Pulmonary fibrosis.

Publication types

  • Case Reports

MeSH terms

  • Aged
  • Carcinoma / diagnosis
  • Carcinoma / drug therapy
  • Endothelium, Vascular / drug effects
  • Endothelium, Vascular / injuries
  • Glomerular Mesangium / blood supply
  • Glomerular Mesangium / drug effects
  • Glomerular Mesangium / injuries
  • Humans
  • Hyperaldosteronism / drug therapy
  • Idiopathic Pulmonary Fibrosis / drug therapy*
  • Indoles / administration & dosage
  • Indoles / adverse effects*
  • Indoles / therapeutic use
  • Kidney / blood supply
  • Kidney / drug effects
  • Kidney Diseases / chemically induced*
  • Kidney Diseases / pathology
  • Lung Neoplasms / pathology
  • Male
  • Protein Kinase Inhibitors / administration & dosage
  • Protein Kinase Inhibitors / adverse effects*
  • Protein Kinase Inhibitors / therapeutic use
  • Proteinuria / chemically induced*
  • Receptors, Fibroblast Growth Factor / drug effects
  • Receptors, Platelet-Derived Growth Factor / drug effects
  • Receptors, Vascular Endothelial Growth Factor / drug effects
  • Thrombotic Microangiopathies / chemically induced
  • Thrombotic Microangiopathies / diagnosis
  • Withholding Treatment

Substances

  • Indoles
  • Protein Kinase Inhibitors
  • Receptors, Fibroblast Growth Factor
  • Receptors, Platelet-Derived Growth Factor
  • Receptors, Vascular Endothelial Growth Factor
  • nintedanib