Oral dosing of Recombinant Methioninase Is Associated With a 70% Drop in PSA in a Patient With Bone-metastatic Prostate Cancer and 50% Reduction in Circulating Methionine in a High-stage Ovarian Cancer Patient

Anticancer Res. 2020 May;40(5):2813-2819. doi: 10.21873/anticanres.14254.

Abstract

Background/aim: Methionine addiction is a general and fundamental hallmark of cancer. Methionine addiction can be targeted by methionine restriction (MR). Our laboratory has studied methionine addiction in cancer and MR for almost 50 years. The present study describes oral recombinant methioninase (o-rMETase), as a supplement, to induce MR in cancer patients.

Patients and methods: One patient, a 67-year-old female with high-stage ovarian cancer took o-rMETase twice a day at 250 units per dose for approximately one month. A second patient, a 76-year-old male with bone-metastatic prostate cancer, took o-rMETase twice a day at 250 units per dose during three months.

Results: The first patient's circulating methionine levels decreased 50% within 4 hours of taking 250 units of o-rMETase. The second patient's PSA dropped approximately 70% over 3 months. During this time the patient's hemoglobin increased.

Conclusion: o-rMETase has no side effects and is potentially efficacious. Future studies involving larger cohorts of patients with high-stage cancer are required to determine if o-rMETase, as a supplement, can increase survival and improve the quality of life.

Keywords: Methioninase; PSA; cancer patients; methionine; methionine restriction prostate cancer; oral; ovarian cancer; supplement.

Publication types

  • Case Reports

MeSH terms

  • Administration, Oral
  • Aged
  • Animals
  • Antimetabolites, Antineoplastic / pharmacology
  • Antimetabolites, Antineoplastic / therapeutic use*
  • Bone Neoplasms / pathology
  • Bone Neoplasms / secondary*
  • Carbon-Sulfur Lyases / pharmacology
  • Carbon-Sulfur Lyases / therapeutic use*
  • Female
  • Humans
  • Male
  • Neoplasm Staging
  • Ovarian Neoplasms / drug therapy*
  • Ovarian Neoplasms / pathology
  • Prostate-Specific Antigen / drug effects*
  • Prostatic Neoplasms / drug therapy*
  • Prostatic Neoplasms / pathology
  • Quality of Life

Substances

  • Antimetabolites, Antineoplastic
  • Prostate-Specific Antigen
  • Carbon-Sulfur Lyases
  • L-methionine gamma-lyase