Development of A MERS-CoV Replicon Cell Line for Antiviral Screening

Virol Sin. 2021 Aug;36(4):730-735. doi: 10.1007/s12250-020-00341-z. Epub 2021 Feb 22.

Abstract

Middle East respiratory syndrome coronavirus (MERS-CoV) is the causative agent of a severe respiratory disease with a high mortality of ~ 35%. The lack of approved treatments for MERS-CoV infection underscores the need for a user-friendly system for rapid drug screening. In this study, we constructed a MERS-CoV replicon containing the Renilla luciferase (Rluc) reporter gene and a stable luciferase replicon-carrying cell line. Using this cell line, we showed that MERS-CoV replication was inhibited by combined application of lopinavir and ritonavir, indicating that this cell line can be used to screen inhibitors of MERS-CoV replication. Importantly, the MERS-replicon cell line can be used for high-throughput screening of antiviral drugs without the need for live virus handling, providing an effective and safe tool for the discovery of antiviral drugs against MERS-CoV.

Keywords: Antiviral screening; Luciferase reporter gene; Middle East respiratory syndrome coronavirus (MERS-CoV); Replicon cell line.

MeSH terms

  • Antiviral Agents* / pharmacology
  • Cell Line*
  • Coronavirus Infections / drug therapy
  • Drug Evaluation, Preclinical*
  • Humans
  • Lopinavir / therapeutic use
  • Middle East Respiratory Syndrome Coronavirus* / genetics
  • Replicon

Substances

  • Antiviral Agents
  • Lopinavir