Mitohormesis reprogrammes macrophage metabolism to enforce tolerance

Nat Metab. 2021 May;3(5):618-635. doi: 10.1038/s42255-021-00392-w. Epub 2021 May 20.

Abstract

Macrophages generate mitochondrial reactive oxygen species and mitochondrial reactive electrophilic species as antimicrobials during Toll-like receptor (TLR)-dependent inflammatory responses. Whether mitochondrial stress caused by these molecules impacts macrophage function is unknown. Here, we demonstrate that both pharmacologically driven and lipopolysaccharide (LPS)-driven mitochondrial stress in macrophages triggers a stress response called mitohormesis. LPS-driven mitohormetic stress adaptations occur as macrophages transition from an LPS-responsive to LPS-tolerant state wherein stimulus-induced pro-inflammatory gene transcription is impaired, suggesting tolerance is a product of mitohormesis. Indeed, like LPS, hydroxyoestrogen-triggered mitohormesis suppresses mitochondrial oxidative metabolism and acetyl-CoA production needed for histone acetylation and pro-inflammatory gene transcription, and is sufficient to enforce an LPS-tolerant state. Thus, mitochondrial reactive oxygen species and mitochondrial reactive electrophilic species are TLR-dependent signalling molecules that trigger mitohormesis as a negative feedback mechanism to restrain inflammation via tolerance. Moreover, bypassing TLR signalling and pharmacologically triggering mitohormesis represents a new anti-inflammatory strategy that co-opts this stress response to impair epigenetic support of pro-inflammatory gene transcription by mitochondria.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetyl Coenzyme A / metabolism
  • Anti-Inflammatory Agents / pharmacology
  • Cellular Reprogramming*
  • Energy Metabolism*
  • Estrogens / metabolism
  • Gene Expression Regulation
  • Immune Tolerance*
  • Lipopolysaccharides / immunology
  • Macrophage Activation
  • Macrophages / immunology*
  • Macrophages / metabolism*
  • Mitochondria / metabolism*
  • Models, Biological
  • Reactive Oxygen Species / metabolism
  • Stress, Physiological

Substances

  • Anti-Inflammatory Agents
  • Estrogens
  • Lipopolysaccharides
  • Reactive Oxygen Species
  • Acetyl Coenzyme A