The NF-κB Transcriptional Footprint Is Essential for SARS-CoV-2 Replication

J Virol. 2021 Nov 9;95(23):e0125721. doi: 10.1128/JVI.01257-21. Epub 2021 Sep 15.

Abstract

SARS-CoV-2, the etiological agent of COVID-19, is characterized by a delay in type I interferon (IFN-I)-mediated antiviral defenses alongside robust cytokine production. Here, we investigate the underlying molecular basis for this imbalance and implicate virus-mediated activation of NF-κB in the absence of other canonical IFN-I-related transcription factors. Epigenetic and single-cell transcriptomic analyses show a selective NF-κB signature that was most prominent in infected cells. Disruption of NF-κB signaling through the silencing of the NF-κB transcription factor p65 or p50 resulted in loss of virus replication that was rescued upon reconstitution. These findings could be further corroborated with the use of NF-κB inhibitors, which reduced SARS-CoV-2 replication in vitro. These data suggest that the robust cytokine production in response to SARS-CoV-2, despite a diminished IFN-I response, is the product of a dependency on NF-κB for viral replication. IMPORTANCE The COVID-19 pandemic has caused significant mortality and morbidity around the world. Although effective vaccines have been developed, large parts of the world remain unvaccinated while new SARS-CoV-2 variants keep emerging. Furthermore, despite extensive efforts and large-scale drug screenings, no fully effective antiviral treatment options have been discovered yet. Therefore, it is of the utmost importance to gain a better understanding of essential factors driving SARS-CoV-2 replication to be able to develop novel approaches to target SARS-CoV-2 biology.

Keywords: NF-κB; SARS-CoV-2.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • A549 Cells
  • Animals
  • COVID-19 / metabolism*
  • COVID-19 / virology
  • Chlorocebus aethiops
  • Cytokines / metabolism*
  • Epigenomics
  • Gene Expression Regulation
  • HEK293 Cells
  • HeLa Cells
  • Host Microbial Interactions
  • Humans
  • Interferon Type I / metabolism*
  • SARS-CoV-2*
  • Signal Transduction
  • Single-Cell Analysis
  • Transcription Factor RelA / antagonists & inhibitors
  • Transcription Factor RelA / genetics
  • Transcription Factor RelA / metabolism*
  • Transcription Factors / metabolism
  • Transcriptome*
  • Vero Cells
  • Virus Replication*

Substances

  • Cytokines
  • Interferon Type I
  • RELA protein, human
  • Transcription Factor RelA
  • Transcription Factors