Resveratrol protects against myocardial ischemia-reperfusion injury via attenuating ferroptosis

Gene. 2022 Jan 15:808:145968. doi: 10.1016/j.gene.2021.145968. Epub 2021 Sep 14.

Abstract

Resveratrol (Res) is a polyphenol with a variety of biological activities. However, whether Res can prevent myocardial ischemia-reperfusion (I/R) injury is not yet known. This study aimed to investigate the protective effect of Res on myocardial I/R injury and to explore its potential mechanism. H9c2 cells were used for the in vitro experiments and oxygen-glucose deprivation/reoxygenation (OGD/R) model was established. Rats were ligated and perfused by the left anterior descending branch with or without Res (50 mg/kg·bw) for 14 days.The higher level of oxidative stress and Fe2+ content was observed in OGD/R-induced H9c2 cells than that of normal cells. OGD/R-induced H9c2 cells showed increased ferroptosis, mainly by reducing the expression of glutathione peroxidase 4 (GPX4) and ferritin heavy chain 1 (FTH1), but enhancing the expression of transferrin receptor 1 (TfR1). Both in vivo and in vitro experiments indicated that Res reduced the level of oxidative stress and Fe2 + content. In addition, Res inhibited ferroptosis, decreased TfR1 expression, and increased the expressions of FTH1 and GPX4 in OGD/R-induced H9c2 cells and I/R rats. Moreover, we found that Res inhibited ferroptosis by the regulation of ubiquity specific peptidase 19 (USP19)-Beclin1 autophagy. Res protects against myocardial I/R injury via reducing oxidative stress and attenuating ferroptosis. Res could be a potential agent to the prevention of myocardial I/R injury.

Keywords: Autophagy; Ferroptosis; Myocardial ischemia-reperfusion; Resveratrol; Ubiquitination.

MeSH terms

  • Animals
  • Apoptosis / drug effects
  • Autophagy / drug effects
  • Cell Line
  • Cell Survival / drug effects
  • Ferroptosis / drug effects*
  • Ferroptosis / physiology
  • Glucose / metabolism
  • Heart / drug effects
  • Male
  • Myocardial Reperfusion Injury / metabolism
  • Myocardial Reperfusion Injury / prevention & control
  • Myocardium / metabolism
  • Myocytes, Cardiac / metabolism
  • Oxidative Stress / drug effects
  • Oxygen / metabolism
  • Protective Agents / pharmacology
  • Rats
  • Rats, Sprague-Dawley
  • Reperfusion Injury / drug therapy*
  • Reperfusion Injury / metabolism
  • Resveratrol / metabolism
  • Resveratrol / pharmacology*
  • Signal Transduction / drug effects

Substances

  • Protective Agents
  • Glucose
  • Resveratrol
  • Oxygen