Platelet Inhibition by Low-Dose Acetylsalicylic Acid Reduces Neuroinflammation in an Animal Model of Multiple Sclerosis

Int J Mol Sci. 2021 Sep 14;22(18):9915. doi: 10.3390/ijms22189915.

Abstract

Aside from the established immune-mediated etiology of multiple sclerosis (MS), compelling evidence implicates platelets as important players in disease pathogenesis. Specifically, numerous studies have highlighted that activated platelets promote the central nervous system (CNS)-directed adaptive immune response early in the disease course. Platelets, therefore, present a novel opportunity for modulating the neuroinflammatory process that characterizes MS. We hypothesized that the well-known antiplatelet agent acetylsalicylic acid (ASA) could inhibit neuroinflammation by affecting platelets if applied at low-dose and investigated its effect during experimental autoimmune encephalomyelitis (EAE) as a model to study MS. We found that oral administration of low-dose ASA alleviates symptoms of EAE accompanied by reduced inflammatory infiltrates and less extensive demyelination. Remarkably, the percentage of CNS-infiltrated CD4+ T cells, the major drivers of neuroinflammation, was decreased to 40.98 ± 3.28% in ASA-treated mice compared to 56.11 ± 1.46% in control animals at the disease maximum as revealed by flow cytometry. More interestingly, plasma levels of thromboxane A2 were decreased, while concentrations of platelet factor 4 and glycoprotein VI were not affected by low-dose ASA treatment. Overall, we demonstrate that low-dose ASA could ameliorate the platelet-dependent neuroinflammatory response in vivo, thus indicating a potential treatment approach for MS.

Keywords: acetylsalicylic acid; experimental autoimmune encephalomyelitis; glycoprotein VI; multiple sclerosis; platelet factor 4; platelets; thromboxane.

MeSH terms

  • Animals
  • Aspirin / administration & dosage
  • Aspirin / pharmacology*
  • Aspirin / therapeutic use
  • Blood Platelets / drug effects
  • Blood Platelets / pathology*
  • Brain / pathology*
  • CD4-Positive T-Lymphocytes / drug effects
  • CD4-Positive T-Lymphocytes / immunology
  • Disease Models, Animal
  • Dose-Response Relationship, Drug
  • Encephalomyelitis, Autoimmune, Experimental / drug therapy
  • Encephalomyelitis, Autoimmune, Experimental / pathology
  • Inflammation / immunology
  • Inflammation / pathology*
  • Mice
  • Mice, Inbred C57BL
  • Multiple Sclerosis / blood*
  • Multiple Sclerosis / immunology
  • Multiple Sclerosis / pathology*
  • Platelet Aggregation Inhibitors / pharmacology*
  • Thromboxane A2 / biosynthesis

Substances

  • Platelet Aggregation Inhibitors
  • Thromboxane A2
  • Aspirin