Real-world ibrutinib dose reductions, holds and discontinuations in chronic lymphocytic leukemia

Future Oncol. 2021 Dec;17(35):4959-4969. doi: 10.2217/fon-2021-0964. Epub 2021 Nov 16.

Abstract

Aim: A retrospective chart review of ibrutinib-treated patients with chronic lymphocytic leukemia (CLL) was conducted. Patients & methods: Adults with CLL who initiated ibrutinib were followed for ≥6 months (n = 180). Results: Twenty-five percent of first-line ibrutinib patients experienced ≥1 dose reduction, mainly due to adverse events (AEs; 79%). Treatment discontinuations and dose holds occurred in 20 and 34% of patients, respectively, most commonly due to AEs (73 and 74%). Approximately one-quarter of relapsed/refractory ibrutinib patients experienced ≥1 dose reduction, mainly due to AEs (88%). Treatment discontinuation and dose holds occurred in 40% of patients (58 and 76% due to AEs, respectively). Conclusion: Dose reductions, holds and discontinuations were frequent in patients with CLL receiving ibrutinib in routine clinical practice.

Keywords: chronic lymphocytic leukemia; discontinuation; dose holds; dose reductions; ibrutinib; real-world evidence.

Plain language summary

Lay abstract Chronic lymphocytic leukemia (CLL) is a cancer that develops from a type of white blood cells called ‘B cells.’ Ibrutinib is a targeted therapy that inhibits the activity of a protein called Bruton’s tyrosine kinase, which plays a key role in CLL. Patients receiving ibrutinib treatment can experience side effects (‘adverse events’). In addition, patients may need to reduce their drug dose (‘dose reductions’) or stop treatment (‘discontinuations’) for a variety of reasons. We reviewed patients’ charts to describe dose reductions and discontinuations in ibrutinib-treated patients with CLL. Our results indicate that dose reductions and discontinuations were frequent in patients with CLL receiving ibrutinib in routine clinical practice, and that the most common reason was adverse events.

Publication types

  • Multicenter Study

MeSH terms

  • Adenine / administration & dosage
  • Adenine / adverse effects
  • Adenine / analogs & derivatives*
  • Adult
  • Aged
  • Aged, 80 and over
  • Clinical Decision-Making
  • Disease Management
  • Drug Resistance, Neoplasm
  • Drug Tapering
  • Female
  • Humans
  • Leukemia, Lymphocytic, Chronic, B-Cell / diagnosis
  • Leukemia, Lymphocytic, Chronic, B-Cell / drug therapy*
  • Leukemia, Lymphocytic, Chronic, B-Cell / etiology
  • Male
  • Middle Aged
  • Molecular Targeted Therapy / methods
  • Piperidines / administration & dosage*
  • Piperidines / adverse effects
  • Protein Kinase Inhibitors / administration & dosage*
  • Protein Kinase Inhibitors / adverse effects
  • Recurrence
  • Retrospective Studies
  • Withholding Treatment

Substances

  • Piperidines
  • Protein Kinase Inhibitors
  • ibrutinib
  • Adenine

Grants and funding