Mechanical activation of lung epithelial cells through the ion channel Piezo1 activates the metalloproteinases ADAM10 and ADAM17 and promotes growth factor and adhesion molecule release

Biomater Adv. 2023 Sep:152:213516. doi: 10.1016/j.bioadv.2023.213516. Epub 2023 Jun 12.

Abstract

In the lung, pulmonary epithelial cells undergo mechanical stretching during ventilation. The associated cellular mechanoresponse is still poorly understood at the molecular level. Here, we demonstrate that activation of the mechanosensitive cation channel Piezo1 in a human epithelial cell line (H441) and in primary human lung epithelial cells induces the proteolytic activity of the metalloproteinases ADAM10 and ADAM17 at the plasma membrane. These ADAMs are known to convert cell surface expressed proteins into soluble and thereby play major roles in proliferation, barrier regulation and inflammation. We observed that chemical activation of Piezo1 promotes cleavage of substrates that are specific for either ADAM10 or ADAM17. Activation of Piezo1 also induced the synthesis and ADAM10/17-dependent release of the growth factor amphiregulin (AREG). In addition, junctional adhesion molecule A (JAM-A) was shed in an ADAM10/17-dependent manner resulting in a reduction of cell contacts. Stretching experiments combined with Piezo1 knockdown further demonstrated that mechanical activation promotes shedding via Piezo1. Most importantly, high pressure ventilation of murine lungs increased AREG and JAM-A release into the alveolar space, which was reduced by a Piezo1 inhibitor. Our study provides a novel link between stretch-induced Piezo1 activation and the activation of ADAM10 and ADAM17 in lung epithelium. This may help to understand acute respiratory distress syndrome (ARDS) which is induced by ventilation stress and goes along with perturbed epithelial permeability and release of growth factors.

Keywords: Cell junctions; Epithelial lung cells; Ion channel; Mechanotransduction; Metalloproteinase; Shedding; Stretch.

MeSH terms

  • ADAM10 Protein / genetics
  • ADAM10 Protein / metabolism
  • ADAM17 Protein / genetics
  • ADAM17 Protein / metabolism
  • Amyloid Precursor Protein Secretases* / genetics
  • Amyloid Precursor Protein Secretases* / metabolism
  • Animals
  • Epithelial Cells / metabolism
  • Humans
  • Intercellular Signaling Peptides and Proteins / genetics
  • Intercellular Signaling Peptides and Proteins / metabolism
  • Ion Channels / metabolism
  • Lung* / metabolism
  • Membrane Proteins / genetics
  • Membrane Proteins / metabolism
  • Metalloproteases / metabolism
  • Mice

Substances

  • Amyloid Precursor Protein Secretases
  • ADAM10 Protein
  • Membrane Proteins
  • Ion Channels
  • Intercellular Signaling Peptides and Proteins
  • Metalloproteases
  • ADAM10 protein, human
  • ADAM17 protein, human
  • ADAM17 Protein
  • Piezo1 protein, mouse