Self-Assembling Peptides with Insulin-Like Growth Factor Mimicry

ACS Appl Mater Interfaces. 2024 Jan 10;16(1):364-375. doi: 10.1021/acsami.3c15660. Epub 2023 Dec 25.

Abstract

Growth factor (GF) mimicry involves recapitulating the signaling of larger molecules or cells. Although GF mimicry holds considerable promise in tissue engineering and drug design applications, difficulties in targeting the signaling molecule to the site of delivery and dissociation of mimicking peptides from their target receptors continue to limit its clinical application. To address these challenges, we utilized a self-assembling peptide (SAP) platform to generate synthetic insulin-like growth factor (IGF)-signaling, self-assembling GFs. Our peptide hydrogels are biocompatible and bind target IGF receptors in a dose-dependent fashion, activate proangiogenic signaling, and facilitate formation of angiogenic microtubules in vitro. Furthermore, infiltrated hydrogels are stable for weeks to months. We conclude that the enhanced targeting and long-term stability of our SAP/GF mimicry implants may improve the efficacy and safety of future GF mimic therapeutics.

Keywords: growth factor mimicry; insulin-like growth factor; receptor binding; self-assembly; tissue engineering.

MeSH terms

  • Hydrogels / chemistry
  • Insulin-Like Peptides*
  • Intercellular Signaling Peptides and Proteins
  • Peptides* / chemistry
  • Tissue Engineering

Substances

  • Insulin-Like Peptides
  • Peptides
  • Intercellular Signaling Peptides and Proteins
  • Hydrogels