Pharmacotherapies for multidrug-resistant gram-positive infections: current options and beyond

Expert Opin Pharmacother. 2024 Jun;25(8):1027-1037. doi: 10.1080/14656566.2024.2367003. Epub 2024 Jun 13.

Abstract

Introduction: Infections due to multidrug-resistant organisms (MDRO) are a serious concern for public health with high morbidity and mortality. Though many antibiotics have been introduced to manage these infections, there are remaining concerns regarding the optimal management of Gram-positive MDROs.

Areas covered: A literature search on the PubMed/Medline database was conducted. We applied no language and time limits for the search strategy. In this narrative review, we discuss the current options for managing Gram-positive MDROs as well as non-traditional antibacterial agents in development.

Expert opinion: Despite their introduction more than 70 years ago, glycopeptides are still the cornerstone in treating Gram-positive infections: all registrative studies of new antibiotics have glycopeptides as control; these studies are designed as not inferior studies, therefore it is almost impossible to give recommendations other than the use of glycopeptides in the treatment of Gram-positive infections. The best evidence on treatments different from glycopeptides comes from post-hoc analysis and meta-analysis. Non-traditional antibacterial agents are being studied to aid in short and effective antibiotic therapies. The use of non-traditional antibacterial agents is not restricted to replacing traditional antibacterial agents with alternative therapies; instead, they should be used in combination with antibiotic therapies.

Keywords: Multidrug-resistant organisms; anti-Gram-positive antibiotics; methicillin-resistant-staphylococcus aureus; penicillin-non-susceptible streptococcus pneumoniae; vancomycin-resistant enterococcus faecium.

Publication types

  • Review

MeSH terms

  • Animals
  • Anti-Bacterial Agents* / pharmacology
  • Anti-Bacterial Agents* / therapeutic use
  • Drug Development
  • Drug Resistance, Multiple, Bacterial*
  • Glycopeptides* / therapeutic use
  • Gram-Positive Bacteria* / drug effects
  • Gram-Positive Bacterial Infections* / drug therapy
  • Gram-Positive Bacterial Infections* / microbiology
  • Humans

Substances

  • Anti-Bacterial Agents
  • Glycopeptides