Reversible acetylation of HDAC8 regulates cell cycle

EMBO Rep. 2024 Sep;25(9):3925-3943. doi: 10.1038/s44319-024-00210-w. Epub 2024 Jul 23.

Abstract

HDAC8, a member of class I HDACs, plays a pivotal role in cell cycle regulation by deacetylating the cohesin subunit SMC3. While cyclins and CDKs are well-established cell cycle regulators, our knowledge of other regulators remains limited. Here we reveal the acetylation of K202 in HDAC8 as a key cell cycle regulator responsive to stress. K202 acetylation in HDAC8, primarily catalyzed by Tip60, restricts HDAC8 activity, leading to increased SMC3 acetylation and cell cycle arrest. Furthermore, cells expressing the mutant form of HDAC8 mimicking K202 acetylation display significant alterations in gene expression, potentially linked to changes in 3D genome structure, including enhanced chromatid loop interactions. K202 acetylation impairs cell cycle progression by disrupting the expression of cell cycle-related genes and sister chromatid cohesion, resulting in G2/M phase arrest. These findings indicate the reversible acetylation of HDAC8 as a cell cycle regulator, expanding our understanding of stress-responsive cell cycle dynamics.

Keywords: 3D Genome Structure; Acetylation; Cell Cycle; HDAC8; Sister Chromatid Cohesion.

MeSH terms

  • Acetylation
  • Cell Cycle Proteins* / genetics
  • Cell Cycle Proteins* / metabolism
  • Cell Cycle* / genetics
  • Chondroitin Sulfate Proteoglycans
  • Chromosomal Proteins, Non-Histone* / genetics
  • Chromosomal Proteins, Non-Histone* / metabolism
  • Histone Acetyltransferases / genetics
  • Histone Acetyltransferases / metabolism
  • Histone Deacetylases* / genetics
  • Histone Deacetylases* / metabolism
  • Humans
  • Lysine Acetyltransferase 5 / genetics
  • Lysine Acetyltransferase 5 / metabolism
  • Repressor Proteins* / genetics
  • Repressor Proteins* / metabolism

Substances

  • Histone Deacetylases
  • HDAC8 protein, human
  • Cell Cycle Proteins
  • Chromosomal Proteins, Non-Histone
  • Repressor Proteins
  • Lysine Acetyltransferase 5
  • SMC3 protein, human
  • KAT5 protein, human
  • Histone Acetyltransferases
  • Chondroitin Sulfate Proteoglycans