The triglyceride-synthesizing enzyme diacylglycerol acyltransferase 2 modulates the formation of the hepatitis C virus replication organelle

PLoS Pathog. 2024 Sep 6;20(9):e1012509. doi: 10.1371/journal.ppat.1012509. eCollection 2024 Sep.

Abstract

The replication organelle of hepatitis C virus (HCV), called membranous web, is derived from the endoplasmic reticulum (ER) and mainly comprises double membrane vesicles (DMVs) that concentrate the viral replication complexes. It also tightly associates with lipid droplets (LDs), which are essential for virion morphogenesis. In particular acyl-CoA:diacylglycerol acyltransferase 1 (DGAT1), a rate-limiting enzyme in triglyceride synthesis, promotes early steps of virus assembly. The close proximity between ER membranes, DMVs and LDs therefore permits the efficient coordination of the HCV replication cycle. Here, we demonstrate that exaggerated LD accumulation due to the excessive expression of the DGAT1 isozyme, DGAT2, dramatically impairs the formation of the HCV membranous web. This effect depended on the enzymatic activity and ER association of DGAT2, whereas the mere LD accumulation was not sufficient to hamper HCV RNA replication. Our lipidomics data indicate that both HCV infection and DGAT2 overexpression induced membrane lipid biogenesis and markedly increased phospholipids with long chain polyunsaturated fatty acids, suggesting a dual use of these lipids and their possible competition for LD and DMV biogenesis. On the other hand, overexpression of DGAT2 depleted specific phospholipids, particularly oleyl fatty acyl chain-containing phosphatidylcholines, which, in contrast, are increased in HCV-infected cells and likely essential for viral infection. In conclusion, our results indicate that lipid exchanges occurring during LD biogenesis regulate the composition of intracellular membranes and thereby affect the formation of the HCV replication organelle. The potent antiviral effect observed in our DGAT2 overexpression system unveils lipid flux that may be relevant in the context of steatohepatitis, a hallmark of HCV infection, but also in physiological conditions, locally in specific subdomains of the ER membrane. Thus, LD formation mediated by DGAT1 and DGAT2 might participate in the spatial compartmentalization of HCV replication and assembly factories within the membranous web.

MeSH terms

  • Diacylglycerol O-Acyltransferase* / genetics
  • Diacylglycerol O-Acyltransferase* / metabolism
  • Endoplasmic Reticulum* / metabolism
  • Endoplasmic Reticulum* / virology
  • Hepacivirus* / physiology
  • Hepatitis C / metabolism
  • Hepatitis C / virology
  • Humans
  • Lipid Droplets / metabolism
  • Lipid Droplets / virology
  • Triglycerides* / metabolism
  • Virus Replication* / physiology

Substances

  • Diacylglycerol O-Acyltransferase
  • DGAT2 protein, human
  • Triglycerides
  • DGAT1 protein, human

Grants and funding

This work was funded by the Deutsche Forschungsgemeinschaft (DFG, German Research Foundation https://www.dfg.de/en/): Project number 417852234 (https://gepris.dfg.de/gepris/projekt/417852234) to G.V. G.V. was further supported by the Leibniz ScienceCampus InterACt, which is funded by the Leibniz Association and the BWFGB Hamburg (W75/2022 InterACt and "Hamburg- X Infektionsforschung”). T.P. Received funding from the Deutsche Forschungsgemeinschaft (DFG, German Research Foundation) under Germany's Excellence Strategy - EXC 2155 - project number 390874280 (https://gepris-extern.dfg.de/gepris/projekt/390874280) and under the SFB900 project A6 - project number 158989968 (https://gepris.dfg.de/gepris/projekt/178926377). The funders had no role in study design, data collection and analysis, decision to publish, or preparation of the manuscript.