Nine months of bedaquiline, linezolid, levofloxacin, clofazimine, and cycloserine chemotherapy for rifampicin/multidrug-resistant tuberculosis: a multicenter, randomized, open-label non-inferiority trial in China

BMC Med. 2024 Sep 19;22(1):401. doi: 10.1186/s12916-024-03633-3.

Abstract

Background: We concurrently developed a prospective study to assess clinical outcomes among patients receiving 9-month bedaquiline (BDQ)-containing regimens, aiming to provide valuable data on the use of this short-course regimen in China.

Methods: This open-label, randomized, controlled, multicenter, non-inferiority trial was conducted at sixteen hospitals, and enrolled participants aged 18 years and older with pulmonary rifampicin/multidrug tuberculosis. Participants were randomly assigned, in a 1:1 ratio. Individuals within the standard-regimen group received 6 months of BDQ, linezolid, levofloxacin, clofazimine, and cycloserine plus 12 months of levofloxacin, and any three potentially effective drugs from clofazimine, cycloserine pyrazinamide, ethambutol and protionamide, whereas individuals within shorter-regimen group received 9 months of BDQ, linezolid, levofloxacin, clofazimine and cycloserine. The primary outcome was the percentage of participants with a composite unfavorable outcome (treatment failure, death, treatment discontinuation, or loss to follow-up) by the end of the treatment course after randomization in the modified intention-to-treat population. The noninferiority margin was 10%. This trial was registered with www.chictr.org.cn , ChiCTR2000029012.

Results: Between Jan 1, 2020, and Dec 31, 2023, 264 were screened and randomly assigned, 132 of 264 participants were assigned to the standard-regimen group and 132 were assigned to the shorter-regimen. Thirty-three (12.55%) of 264 participants were excluded from the modified intention-to-treat analysis. As a result, 231 participants were included in the modified intention-to-treat analysis (116 in the standard-regimen group and 115 in the shorter-regimen group).In the modified intention-to-treat population, unfavorable outcomes were reported in 19 (16.5%) of 115 participants for whom the outcome was assessable in the shorter-regimen group and 26 (22.4%) of 116 participants in the standard care group (risk difference 5.9 percentage points (97.5% CI - 5.8 to 17.5)). One death was reported in the standard-regimen group. The incidence of QTcF prolongation in the shorter-regimen group (22.6%, 26/115) was similar to the standard-regimen group (24.1%, 28/116).

Conclusions: The 9-month, all-oral regimen is safe and efficacious for the treatment of pulmonary rifampicin/multidrug-resistant tuberculosis. The high incidence of QTc prolongation associated with the use of BDQ highlights the urgent need of routine electrocardiogram monitoring under treatment with BDQ-containing regimens in the Chinese population.

Keywords: Efficacy; Multidrug-resistant; RCT trial; Safety; Tuberculosis.

Publication types

  • Multicenter Study
  • Randomized Controlled Trial

MeSH terms

  • Adult
  • Aged
  • Antitubercular Agents* / administration & dosage
  • Antitubercular Agents* / therapeutic use
  • China / epidemiology
  • Clofazimine* / administration & dosage
  • Clofazimine* / therapeutic use
  • Cycloserine* / administration & dosage
  • Cycloserine* / therapeutic use
  • Diarylquinolines* / administration & dosage
  • Diarylquinolines* / therapeutic use
  • Drug Therapy, Combination
  • Female
  • Humans
  • Levofloxacin* / administration & dosage
  • Levofloxacin* / therapeutic use
  • Linezolid* / administration & dosage
  • Linezolid* / therapeutic use
  • Male
  • Middle Aged
  • Prospective Studies
  • Rifampin* / administration & dosage
  • Rifampin* / therapeutic use
  • Treatment Outcome
  • Tuberculosis, Multidrug-Resistant* / drug therapy
  • Young Adult

Substances

  • bedaquiline
  • Clofazimine
  • Linezolid
  • Diarylquinolines
  • Cycloserine
  • Levofloxacin
  • Antitubercular Agents
  • Rifampin