The cardioprotective effects of Fruitflow® against Doxorubicin-induced toxicity in rat cardiomyoblast cells H9c2 (2-1) and high-fat diet-induced dyslipidemia and pathological alteration in cardiac tissue of Wistar Albino rats

Biomed Pharmacother. 2024 Nov:180:117607. doi: 10.1016/j.biopha.2024.117607. Epub 2024 Oct 30.

Abstract

Background: Natural compounds offer promising targets for cardioprotection, which could lead to enhanced clinical outcomes. We aimed to determine the cardioprotective effects of Fruitflow®, a water-soluble tomato extract known for its anti-platelet effects in doxorubicin-induced toxicity in rat cardiomyoblast cell line pathological alteration in heart tissue of high fat-fed Wistar Albino rats.

Methods: The cardioprotective effect of Fruitflow® was investigated using H9c2 (2-1) cells (rat cardiomyoblast cell line) and high-fat diet-fed Wistar Albino rats. We evaluated morphological changes, cell proliferation, cell migration, antioxidant activity, cell cycle progression, and mitochondrial membrane potential after the Fruitflow® treatment in the Doxorubicin-injured H9c2 (2-1) cell line. We studied lipid profiles, inflammation, oxidative stress, and cardiac function regulatory enzyme activity in the rat model.

Results: Fruitflow® dose-dependently stimulated cell proliferation and migration in Doxorubicin-injured H9c2 (2-1) cells, potentially promoting cardiac regeneration and supporting tissue repair. Fruitflow® modulated the cell cycle, improved mitochondrial function, and reduced oxidative stress. Furthermore, it significantly improved lipid profiles and enzyme activities and reduced inflammation and oxidative stress in high-fat-fed rats. Fruitflow® also modulated the expression of genes involved in cardiac remodeling, mitochondrial biogenesis, inflammation, and vascular function.

Conclusion: Our findings suggest Fruitflow® may have cardioprotective effects, making it a potential treatment option for cardiac ailments. Larger-scale clinical trials were recommended further to determine the efficacy and safety of Fruitflow® as a potential therapeutic agent for cardiac diseases, potentially in combination with other cardioprotective medications.

Keywords: Cardiotoxicity; Doxorubicin; Fruitflow®; H9c2 (2-1) cells; High-fat diet.

MeSH terms

  • Animals
  • Antioxidants / pharmacology
  • Cardiotonic Agents / pharmacology
  • Cardiotoxicity
  • Cell Line
  • Cell Movement / drug effects
  • Cell Proliferation* / drug effects
  • Diet, High-Fat* / adverse effects
  • Doxorubicin* / adverse effects
  • Doxorubicin* / toxicity
  • Dyslipidemias* / drug therapy
  • Male
  • Membrane Potential, Mitochondrial / drug effects
  • Myoblasts, Cardiac / drug effects
  • Myoblasts, Cardiac / metabolism
  • Myoblasts, Cardiac / pathology
  • Oxidative Stress* / drug effects
  • Plant Extracts* / pharmacology
  • Rats
  • Rats, Wistar*

Substances

  • Doxorubicin
  • Plant Extracts
  • Cardiotonic Agents
  • Antioxidants