A practical procedure for testing DNA damage in vivo, proposed for a pre-screening of chemical carcinogens

Mutat Res. 1978 Aug;54(1):39-46. doi: 10.1016/0165-1161(78)90133-4.

Abstract

The alkaline elution method was adapted to the evaluation of DNA damage induced in vivo through a practical and reliable microfluorometric procedure, without any need for tissue pre-labeling. The DNA damage induced in vivo by treatment with a single dose of N-nitrosodimethylamine (DMNA), N-methyl-N-nitroso-urea (MNU), 1,2-dimethylhydrazine (DMH) or cycasin has been detected in different organs of mice or rats. The results obtained are rather consistent with the organotropism of these carcinogens, and show a satisfactory dose dependent of DNA damage. DMH and cycasin, both negative in the Ames' Salmonella/microsome mutagenicity test, are clearly positive with in vivo DNA damage/alkaline elution assay. This latter method, complemented with other short-term tests, may play a useful role in the pre-screening of chemical carcinogens.

MeSH terms

  • Animals
  • Brain / metabolism
  • Carcinogens / pharmacology*
  • Cycasin / pharmacology
  • DNA / metabolism*
  • Dimethylhydrazines / pharmacology
  • Dimethylnitrosamine / pharmacology
  • Drug Evaluation, Preclinical / methods*
  • Fluorometry / methods*
  • Kidney / metabolism
  • Liver / metabolism
  • Lung / metabolism
  • Methylnitrosourea / pharmacology
  • Mice
  • Mice, Inbred BALB C
  • Rats

Substances

  • Carcinogens
  • Dimethylhydrazines
  • Methylnitrosourea
  • DNA
  • Cycasin
  • Dimethylnitrosamine