Differential influence of arachidonic vs. eicosapentaenoic acid on experimental pulmonary hypertension

Am J Physiol. 1995 Jun;268(6 Pt 2):H2252-9. doi: 10.1152/ajpheart.1995.268.6.H2252.

Abstract

The impact of the 2- and 3-series prostanoid precursors arachidonic acid (AA) and eicosapentaenoic acid (EPA) on experimental pulmonary hypertension was investigated. The model of buffer-perfused rabbit lungs was stimulated by infusion of Escherichia coli hemolysin (HlyA), which is known to provoke sustained thromboxane (Tx)-mediated pulmonary hypertension. Release of di- and trienoic Tx into the recirculating perfusate was quantified by a post-high-performance liquid chromatography enzyme-linked immunosorbent assay technique. HlyA at 0.08 hemolytic unit/ml caused a sustained rise in pulmonary arterial pressure (PAP; maximum increase 14 +/- 2 mmHg) accompanied by progressive TxB2 liberation (maximum perfusate concn 33 +/- 4 pg/ml, baseline < 2 pg/ml). Between 5 and 30 nM, AA provoked a transient monophasic rise in PAP (maximum pressor response 1.5-15 mmHg) and concomitant TxB2 release (peak concn 2-30 pg/ml). Simultaneous administration of HlyA and AA exhibited additive effects with regard to mediator release and pressor responses. EPA at 200-2,000 nM caused a transient rise in PAP similar to that provoked by 5-30 nM AA (maximum pressor response 3-18 mmHg). This was accompanied by liberation of TxB2 (peak concn 16 +/- 5 and 28 +/- 4 pg/ml after 1,000 and 2,000 nM EPA) and TxB3 (peak concn 9 +/- 4 and 30 +/- 3 pg/ml). Combined application of HlyA and EPA resulted in approximate addition of the TxB2 release reaction to each single compound, and TxB3 liberation more than doubled (maximum concn 59 +/- 12 pg/ml). The pressor responses to HlyA-EPA (200-2,000 nM) did not, however, surpass those to HlyA-AA (5-30 nM).(ABSTRACT TRUNCATED AT 250 WORDS)

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Arachidonic Acid / pharmacology*
  • Disease Models, Animal
  • Dose-Response Relationship, Drug
  • Eicosapentaenoic Acid / pharmacology*
  • Escherichia coli
  • Female
  • Hemolysin Proteins / toxicity
  • Hypertension, Pulmonary / physiopathology*
  • Male
  • Potassium / blood
  • Pulmonary Artery / drug effects
  • Pulmonary Artery / physiopathology*
  • Pulmonary Wedge Pressure / drug effects
  • Pulmonary Wedge Pressure / physiology*
  • Rabbits
  • Thromboxane B2 / analogs & derivatives
  • Thromboxane B2 / metabolism
  • Thromboxanes* / analogs & derivatives*

Substances

  • Hemolysin Proteins
  • Thromboxanes
  • Arachidonic Acid
  • Thromboxane B2
  • Eicosapentaenoic Acid
  • Potassium
  • thromboxane B3