Three months of octreotide treatment decreases gastric acid secretion and argyrophil cell density in patients with Zollinger-Ellison syndrome and antral G-cell hyperfunction

Aliment Pharmacol Ther. 1994 Feb;8(1):95-104. doi: 10.1111/j.1365-2036.1994.tb00165.x.

Abstract

Methods: The effects of three months of treatment with octreotide on gastric acid hypersecretion induced by hypergastrinaemia were investigated in patients with Zollinger-Ellison syndrome (n = 5) or antral G-cell hyperfunction (n = 4). Gastric acid secretion, fasting plasma gastrin concentrations and clinical findings were examined, and a morphometrical analysis of oxyntic endocrine cells was performed.

Results: Administration of octreotide 100 mcg b.d. subcutaneously significantly decreased the volume density of argyrophil cells (P < 0.05) as well as basal and pentagastrin-stimulated acid secretion (P < 0.05). Although partial or complete loss of inhibition was found in most patients after 3 months, gastrin levels were decreased during the first 2 months of treatment (P < 0.05). Fundic D-cells were not affected by treatment. Positive correlations were observed between volume density of argyrophil cells and basal acid output (r = 0.65); plasma gastrin and basal acid output (r = 0.74); plasma gastrin concentrations and volume density of argyrophil cells (r = 0.80).

Conclusion: These results support the important role of the enterochromaffin-like cell in maintaining acid secretion, and indicate a specific role for octreotide in the therapy of gastric acid hypersecretion associated with hypergastrinaemic diseases.

Publication types

  • Clinical Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Oral
  • Adult
  • Cell Count / drug effects
  • Enterochromaffin Cells / drug effects*
  • Enterochromaffin Cells / pathology
  • Female
  • Gastric Acid / metabolism*
  • Gastrins / blood*
  • Humans
  • Male
  • Middle Aged
  • Octreotide / administration & dosage
  • Octreotide / adverse effects
  • Octreotide / blood
  • Octreotide / therapeutic use*
  • Pyloric Antrum / drug effects*
  • Pyloric Antrum / pathology
  • Somatostatin / metabolism
  • Zollinger-Ellison Syndrome / drug therapy*
  • Zollinger-Ellison Syndrome / metabolism
  • Zollinger-Ellison Syndrome / pathology

Substances

  • Gastrins
  • Somatostatin
  • Octreotide