Characterization of an outward potassium current in canine jejunal circular smooth muscle and its activation by fenamates

J Physiol. 1993 Aug:468:297-310. doi: 10.1113/jphysiol.1993.sp019772.

Abstract

1. A perforated patch clamp technique was used to study an outward potassium current in freshly dissociated circular smooth muscle cells of the canine jejunum. 2. A voltage-dependent outward current was identified which was highly potassium selective, weakly holding voltage sensitive, increased its open probability at -65 mV, and reached unit open probability at +5 mV. 3. Quinidine (0.1-1 mM) and tetraethylammonium ion (TEA) (10-50 mM), blocked the potassium current in a dose-dependent manner. Blockade of the outward potassium current was accompanied by membrane depolarization which reversed on removal of the blocker from the bathing solution. 4. Mefenamic and flufenamic acids, non-steroidal anti-inflammatory agents in the fenamate group, were potent activators of the current. Activation was accompanied by hyperpolarization of the membrane with a mean shift in the membrane voltage of 22 mV. 5. It was concluded that the outward potassium current is a major regulator of the resting membrane voltage in isolated circular smooth muscle cells of the canine jejunum. Fenamates activated this current with potentially profound effects on cellular excitability.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Calcium / pharmacology
  • Dogs
  • Electric Conductivity
  • Female
  • Flufenamic Acid / pharmacology
  • In Vitro Techniques
  • Jejunum / drug effects
  • Jejunum / metabolism*
  • Male
  • Mefenamic Acid / pharmacology
  • Membrane Potentials / drug effects
  • Muscle, Smooth / drug effects
  • Muscle, Smooth / metabolism*
  • Potassium / metabolism*
  • Potassium Channels / drug effects
  • Potassium Channels / metabolism
  • Quinidine / pharmacology
  • Rubidium / pharmacology
  • Tetraethylammonium
  • Tetraethylammonium Compounds / pharmacology

Substances

  • Potassium Channels
  • Tetraethylammonium Compounds
  • Mefenamic Acid
  • Flufenamic Acid
  • Tetraethylammonium
  • Quinidine
  • Rubidium
  • Potassium
  • Calcium