Salivary excretory pattern of testosterone in substitutive therapy with testosterone enanthate

Fertil Steril. 1994 Jan;61(1):125-8. doi: 10.1016/s0015-0282(16)56464-4.

Abstract

Objective: To determine salivary and serum T levels by an RIA method after a single injection of 250 mg IM of commercially available T enanthate.

Design: Research study.

Setting: Patients attended in a hospital environment.

Patients: Sixteen men with secondary hypogonadism.

Interventions: Testosterone enanthate was administered, and salivary samples were taken before the injection. Thereafter, these samples were obtained daily until day 7 and then on alternate days until day 28 after injection. Blood samples were taken previously and after the injection (5 samples during the month).

Main outcome measure: Salivary and serum T.

Results: Salivary T levels rose from 3.46 +/- 3.16 to 13.82 +/- 7.78 ng/100 mL (0.12 +/- 0.11 to 0.48 +/- 0.27 nmol/L) within 24 hours and remained in that range until day 7. From day 9, 7.20 +/- 2.88 ng/100 mL (0.25 +/- 0.10 nmol/L), a progressive decrease of these values was observed until day 14: 5.18 +/- 2.88 ng/100 mL (0.18 +/- 0.10 nmol/L). From day 16 until day 28, salivary concentrations returned to hypogonadal levels.

Conclusion: We conclude that T salivary concentrations may be applied to assess the effectiveness of T substitutive therapy in hypogonadal men and could replace serum in the monitoring of this type of therapy.

MeSH terms

  • Adult
  • Humans
  • Hypogonadism / drug therapy*
  • Injections, Intramuscular
  • Longitudinal Studies
  • Male
  • Middle Aged
  • Radioimmunoassay
  • Salivary Glands / drug effects
  • Salivary Glands / metabolism*
  • Testosterone / administration & dosage
  • Testosterone / analogs & derivatives*
  • Testosterone / blood
  • Testosterone / metabolism*
  • Testosterone / pharmacology
  • Testosterone / therapeutic use
  • Time Factors

Substances

  • Testosterone
  • testosterone enanthate