Pyrophosphate-dependent phosphofructokinase from the amoeba Naegleria fowleri, an AMP-sensitive enzyme

Biochem J. 1993 Jun 15;292 ( Pt 3)(Pt 3):797-803. doi: 10.1042/bj2920797.

Abstract

PPi-dependent phosphofructokinase (PPi-PFK) was detected in extracts of the amoeba Naegleria fowleri, with a specific activity of about 15-30 nmol/min per mg of protein, which was increased about 2-fold by 0.5 mM AMP. PPi-PFK was inactivated upon gel filtration and could be re-activated by incubation at 30 degrees C in the presence of AMP. N. fowleri PPi-PFK was purified more than 1100-fold to near homogeneity with a yield of about 25%. The pure enzyme had a specific activity of 65 mumol/min per mg of protein, and SDS/PAGE analysis showed a single band, of 51 kDa. Size-exclusion chromatography revealed the existence of two forms: a large one (approximately 180 kDa), presumably a tetramer, which was active, and a smaller one (approximately 45 kDa), presumably the monomer, which was inactive, but could be re-activated and converted into the large form by incubation at 30 degrees C in the presence of 0.5 mM AMP. Reactivation was also observed at 30 degrees C in the absence of AMP, particularly at higher enzyme concentration or in the presence of poly(ethylene glycol). Inactivation of the tetrameric enzyme was promoted by 0.25 M potassium thiocyanate. The enzyme displayed Km values of 10 and 15 microM for fructose 6-phosphate and PPi, respectively, in the forward reaction, and of 35 and 590 microM for fructose 1,6-bisphosphate and Pi in the backward reaction. The activity was dependent on the presence of Mg2+. AMP increased Vmax. about 2-fold without changing the affinity for the substrates; its half-maximal effect was observed at 2 microM.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenosine Monophosphate / pharmacology
  • Animals
  • Chromatography, Gel
  • Chromatography, Ion Exchange
  • Detergents / pharmacology
  • Diphosphates / metabolism*
  • Electrophoresis, Polyacrylamide Gel
  • Enzyme Activation
  • Fructosediphosphates / pharmacology
  • Kinetics
  • Macromolecular Substances
  • Molecular Weight
  • Naegleria fowleri / enzymology*
  • Octoxynol
  • Phosphofructokinase-1 / isolation & purification
  • Phosphofructokinase-1 / metabolism*
  • Polyethylene Glycols / pharmacology
  • Spectrophotometry, Ultraviolet
  • Substrate Specificity
  • Thiocyanates / pharmacology

Substances

  • Detergents
  • Diphosphates
  • Fructosediphosphates
  • Macromolecular Substances
  • Thiocyanates
  • Polyethylene Glycols
  • Adenosine Monophosphate
  • fructose 2,6-diphosphate
  • Octoxynol
  • Phosphofructokinase-1
  • potassium thiocyanate