Megakaryocyte growth and development factor stimulates enhanced platelet recovery in mice after bone marrow transplantation

Blood. 1996 Aug 15;88(4):1509-14.

Abstract

Megakaryocyte growth and development factor (MGDF) is a recently characterized ligand for the cell surface receptor mpl. We have evaluated the effects of polyethylene glycollated recombinant human MGDF (PEG-rHuMGDF) on recovery of hematopoietic cells in mice following bone marrow transplantation (BMT) to support lethal irradiation. Mice treated with PEG-rHuMGDF (50 micrograms/kg/d) had accelerated recovery of platelet numbers compared with BMT mice treated with carrier or recombinant human granulocyte colony-stimulating factor (rHuG-CSF, 72 or 200 micrograms/kg/d). In contrast, PEG-rHuMGDF had no effect on white blood cell (WBC) or red blood cell (RBC) recovery. As previously reported, animals treated with rHuG-CSF had an enhanced recovery of WBC but not platelet or RBC levels. Interestingly, BMT receipient mice treated with the combination of PEG-rHuMGDF and rHuG-CSF showed simultaneous enhanced recovery of both leukocytes and platelets. PEGylated rHuMGDF was found to be considerably more potent than non-PEGylated rHuMGDF in this setting. PEG-rHuMGDF is an effective growth factor for enhancing platelet recovery in mice following BMT either alone or in combination with rHuG-CSF. It will be of interest to evaluate in a clinical setting the ratios of PEG-rHuMGDF and rHuG-CSF for simultaneous administration of these factors and accelerated recovery of both leukocytes and platelets.

MeSH terms

  • Animals
  • Blood Platelets / cytology*
  • Bone Marrow Transplantation / pathology*
  • Colony-Stimulating Factors / pharmacology*
  • GPI-Linked Proteins
  • Granulocyte Colony-Stimulating Factor / pharmacology
  • Hematopoiesis / drug effects*
  • Humans
  • Leukocytes / cytology
  • Megakaryocytes / cytology*
  • Membrane Glycoproteins
  • Mesothelin
  • Mice
  • Mice, Inbred C57BL
  • Mice, Inbred DBA
  • Neoplasm Proteins*
  • Polyethylene Glycols*
  • Proteins / pharmacology*
  • Proto-Oncogene Proteins / physiology
  • Radiation Chimera
  • Receptors, Cytokine*
  • Receptors, Thrombopoietin
  • Recombinant Proteins
  • Thrombopoietin / pharmacology*
  • Thrombopoietin / physiology

Substances

  • Colony-Stimulating Factors
  • GPI-Linked Proteins
  • Membrane Glycoproteins
  • Neoplasm Proteins
  • Proteins
  • Proto-Oncogene Proteins
  • Receptors, Cytokine
  • Receptors, Thrombopoietin
  • Recombinant Proteins
  • polyethylene glycol-recombinant human megakaryocyte growth and development factor
  • Granulocyte Colony-Stimulating Factor
  • MPL protein, human
  • Polyethylene Glycols
  • Thrombopoietin
  • Mesothelin