Up-regulation of D3 dopamine receptor mRNA in the nucleus accumbens of human cocaine fatalities

Brain Res Mol Brain Res. 1997 May;45(2):335-9. doi: 10.1016/s0169-328x(97)00025-9.

Abstract

The effects of chronic cocaine use on D3 receptor mRNA expression in the human nucleus accumbens was assessed by reverse transcription-polymerase chain reaction. D3 receptor/cyclophilin mRNA ratios in the nucleus accumbens were increased 6-fold in cocaine overdose victims as compared to age-matched and drug-free control subjects. This finding demonstrates that chronic cocaine exposure leads to adaptive increases in the expression of D3 receptor mRNA in a critical reward center in brain.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Autopsy
  • Cocaine / poisoning*
  • DNA Primers
  • Drug Overdose
  • Humans
  • Nucleus Accumbens / drug effects
  • Nucleus Accumbens / metabolism*
  • Polymerase Chain Reaction
  • RNA, Messenger / biosynthesis
  • Receptors, Dopamine D2 / biosynthesis*
  • Receptors, Dopamine D3
  • Reference Values
  • Transcription, Genetic / drug effects
  • Up-Regulation

Substances

  • DNA Primers
  • DRD3 protein, human
  • RNA, Messenger
  • Receptors, Dopamine D2
  • Receptors, Dopamine D3
  • Cocaine