Selective inhibition of the monosynaptic spinal reflex by a series of hydroxylated alkylaminoindans

J Med Chem. 1977 Nov;20(11):1478-85. doi: 10.1021/jm00221a023.

Abstract

5-Hydroxy-2-piperidino-4,5,6,7-tetrahydroindan (5) and a number of related tetrahydro and dihydro compounds were prepared by selective mono- and dihydroxylation of the dihydro products from the Birch reduction of various alkylaminoalkylindans, tetralins, benzenes, and isoindolines. Some of these compounds showed a remarkably selective inhibition of monosynatpic spinal reflex in the segmental cat preparation.

MeSH terms

  • Animals
  • Cats
  • Decerebrate State
  • Depression, Chemical
  • Electric Stimulation
  • Hydroxylation
  • Indans / chemical synthesis*
  • Indans / pharmacology
  • Indenes / chemical synthesis*
  • Reflex, Monosynaptic / drug effects*
  • Spinal Nerve Roots / drug effects
  • Spinal Nerve Roots / physiology*

Substances

  • Indans
  • Indenes