Binding of the alpha 2 integrin I domain to extracellular matrix ligands: structural and mechanistic differences between collagen and laminin binding

Cell Adhes Commun. 1998 Jun;5(4):273-81. doi: 10.3109/15419069809040297.

Abstract

The alpha 2 beta 1 integrin functions as a cell surface receptor for collagen on some cells and as both a collagen and laminin receptor on a more restricted subset of cell types including endothelial and epithelial cells. The alpha 2 integrin subunit I domain binds collagen in a divalent cation-dependent manner. In contrast, I domain binding to laminin occurs via both divalent cation-dependent and -independent mechanisms. Saturable binding was observed in the presence of either Mn2+ or EDTA, although the extent of binding in Mn2+ was twice that observed in EDTA. Half-maximal binding occurred at about 22 nM I domain in either case. Whereas laminin binding was significantly enhanced by Mn2+, with half-maximal binding occurring at 1.9 mM Mn2+, Mg2+ was much less effective. Deletion of the N-terminal 35 residues of the I domain, including the DXSXS portion of the MIDAS motif, caused a significant diminution of laminin binding activity. Laminin binding by the I domain was significantly inhibited by the alpha 2 beta 1 function-blocking antibody 6F1 in the presence of either EDTA or Mn2+. The non-function-blocking antibody 12F1 had no effect. In contrast to the binding of the alpha 2 integrin I domain to collagen, the laminin binding activity of the I domain was not enhanced by the addition of the first EF hand motif of the integrin.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antibodies, Monoclonal
  • Antigens, CD / chemistry*
  • Antigens, CD / genetics
  • Antigens, CD / metabolism*
  • Cations, Divalent / metabolism
  • Chelating Agents / pharmacology
  • Cloning, Molecular
  • Collagen / metabolism*
  • Edetic Acid / pharmacology
  • Extracellular Space / metabolism*
  • Humans
  • Integrin alpha2
  • Laminin / immunology
  • Laminin / metabolism*
  • Ligands
  • Magnesium / pharmacology
  • Manganese / pharmacology
  • Mutagenesis / physiology
  • Protein Binding / drug effects
  • Protein Binding / physiology
  • Protein Structure, Tertiary

Substances

  • Antibodies, Monoclonal
  • Antigens, CD
  • Cations, Divalent
  • Chelating Agents
  • Integrin alpha2
  • Laminin
  • Ligands
  • Manganese
  • Collagen
  • Edetic Acid
  • Magnesium