Structure of the Ets-1 pointed domain and mitogen-activated protein kinase phosphorylation site

Proc Natl Acad Sci U S A. 1998 Oct 13;95(21):12129-34. doi: 10.1073/pnas.95.21.12129.

Abstract

The Pointed (PNT) domain and an adjacent mitogen-activated protein (MAP) kinase phosphorylation site are defined by sequence conservation among a subset of ets transcription factors and are implicated in two regulatory strategies, protein interactions and posttranslational modifications, respectively. By using NMR, we have determined the structure of a 110-residue fragment of murine Ets-1 that includes the PNT domain and MAP kinase site. The Ets-1 PNT domain forms a monomeric five-helix bundle. The architecture is distinct from that of any known DNA- or protein-binding module, including the helix-loop-helix fold proposed for the PNT domain of the ets protein TEL. The MAP kinase site is in a highly flexible region of both the unphosphorylated and phosphorylated forms of the Ets-1 fragment. Phosphorylation alters neither the structure nor monomeric state of the PNT domain. These results suggest that the Ets-1 PNT domain functions in heterotypic protein interactions and support the possibility that target recognition is coupled to structuring of the MAP kinase site.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Calcium-Calmodulin-Dependent Protein Kinases / metabolism*
  • Magnetic Resonance Spectroscopy
  • Mice
  • Molecular Sequence Data
  • Phosphorylation
  • Protein Conformation
  • Proto-Oncogene Protein c-ets-1
  • Proto-Oncogene Proteins / chemistry
  • Proto-Oncogene Proteins / metabolism*
  • Proto-Oncogene Proteins c-ets
  • Sequence Homology, Amino Acid
  • Transcription Factors / chemistry
  • Transcription Factors / metabolism*

Substances

  • Ets1 protein, mouse
  • Proto-Oncogene Protein c-ets-1
  • Proto-Oncogene Proteins
  • Proto-Oncogene Proteins c-ets
  • Transcription Factors
  • Calcium-Calmodulin-Dependent Protein Kinases

Associated data

  • PDB/1BQV
  • PDB/R1BQVMR