Level and function of epidermal growth factor receptor predict the metastatic potential of human colon carcinoma cells

Clin Cancer Res. 1995 Jan;1(1):19-31.

Abstract

The purpose of this study was to determine whether production of liver metastasis by human colon carcinoma (HCC) cells depends on the response of tumor cells to organ-derived growth factors. HCC cells were isolated from several surgical specimens whose malignant potential differed (Dukes' stage B or D tumors), adapted to grow in culture, and assessed for expression of the epidermal growth factor receptor (EGF-R). Northern blot analyses revealed that highly metastatic HCC cells expressed >5-fold the number of EGF-R mRNA transcripts as low metastatic cells. The level of mRNA correlated with the amount of EGF-R protein as detected by Western blotting, immunohistochemistry, and Scatchard analyses. HCC growth response in vitro to picograms of transforming growth factor alpha was associated with functional cell surface EGF-Rs as determined by receptor tyrosine kinase activity assays. The EGF-R gene was not amplified or rearranged in highly metastatic cells. However, fluorescence in situ hybridization analysis showed that the copy number of chromosome 7 was higher in the highly metastatic cells. HCC cells were selected in vitro for low or high expression of EGF-R. Subsequent to injection into nude mice, only cells with high expression of EGF-R produced a high incidence of liver metastasis. These data demonstrate that expression of EGF-R by HCC cells directly correlates with their ability to produce hepatic metastasis.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Carcinoma, Squamous Cell
  • Cell Division / drug effects
  • Chromosome Mapping
  • Chromosomes, Human, Pair 7
  • Colonic Neoplasms / genetics
  • Colonic Neoplasms / metabolism
  • Colonic Neoplasms / pathology*
  • ErbB Receptors / analysis
  • ErbB Receptors / genetics*
  • ErbB Receptors / metabolism
  • Humans
  • Liver Neoplasms / pathology
  • Liver Neoplasms / secondary*
  • Male
  • Mice
  • Mice, Nude
  • Neoplasm Metastasis*
  • RNA, Messenger / analysis
  • Transcription, Genetic*
  • Transforming Growth Factor alpha / pharmacology
  • Transforming Growth Factor alpha / physiology
  • Transplantation, Heterologous
  • Tumor Cells, Cultured

Substances

  • RNA, Messenger
  • Transforming Growth Factor alpha
  • ErbB Receptors