Analysis of the regulatory phosphorylation site in Acanthamoeba myosin IC by using site-directed mutagenesis

Proc Natl Acad Sci U S A. 1998 Dec 22;95(26):15200-5. doi: 10.1073/pnas.95.26.15200.

Abstract

The actin-activated ATPase activity of Acanthamoeba myosin IC is stimulated 15- to 20-fold by phosphorylation of Ser-329 in the heavy chain. In most myosins, either glutamate or aspartate occupies this position, which lies within a surface loop that forms part of the actomyosin interface. To investigate the apparent need for a negative charge at this site, we mutated Ser-329 to alanine, asparagine, aspartate, or glutamate and coexpressed the Flag-tagged wild-type or mutant heavy chain and light chain in baculovirus-infected insect cells. Recombinant wild-type myosin IC was indistinguishable from myosin IC purified from Acanthamoeba as determined by (i) the dependence of its actin-activated ATPase activity on heavy-chain phosphorylation, (ii) the unusual triphasic dependence of its ATPase activity on the concentration of F-actin, (iii) its Km for ATP, and (iv) its ability to translocate actin filaments. The Ala and Asn mutants had the same low actin-activated ATPase activity as unphosphorylated wild-type myosin IC. The Glu mutant, like the phosphorylated wild-type protein, was 16-fold more active than unphosphorylated wild type, and the Asp mutant was 8-fold more active. The wild-type and mutant proteins had the same Km for ATP. Unphosphorylated wild-type protein and the Ala and Asn mutants were unable to translocate actin filaments, whereas the Glu mutant translocated filaments at the same velocity, and the Asp mutant at 50% the velocity, as phosphorylated wild-type proteins. These results demonstrate that an acidic amino acid can supply the negative charge in the surface loop required for the actin-dependent activities of Acanthamoeba myosin IC in vitro and indicate that the length of the side chain that delivers this charge is important.

MeSH terms

  • Acanthamoeba / metabolism*
  • Actins / metabolism
  • Amino Acid Sequence
  • Amino Acid Substitution
  • Animals
  • Base Sequence
  • Cell Line
  • DNA Primers
  • Isoenzymes / chemistry
  • Isoenzymes / metabolism
  • Kinetics
  • Molecular Sequence Data
  • Mutagenesis, Site-Directed
  • Myosin Heavy Chains / chemistry*
  • Myosin Heavy Chains / metabolism*
  • Myosins / chemistry*
  • Myosins / metabolism*
  • Phosphorylation
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / metabolism
  • Serine
  • Spodoptera
  • Transfection

Substances

  • Actins
  • DNA Primers
  • Isoenzymes
  • Recombinant Proteins
  • Serine
  • Myosin Heavy Chains
  • Myosins

Associated data

  • GENBANK/AF051353