Negri L - Search Results

1

Highly selective fluorescent analogue of the potent delta-opioid receptor antagonist Dmt-Tic.

Balboni G, Salvadori S, Dal Piaz A, Bortolotti F, Argazzi R, Negri L, Lattanzi R, Bryant SD, Jinsmaa Y, Lazarus LH. Balboni G, et al. Among authors: negri l. J Med Chem. 2004 Dec 16;47(26):6541-6. doi: 10.1021/jm040128h. J Med Chem. 2004. PMID: 15588089

2

Potent delta-opioid receptor agonists containing the Dmt-Tic pharmacophore.

Balboni G, Salvadori S, Guerrini R, Negri L, Giannini E, Jinsmaa Y, Bryant SD, Lazarus LH. Balboni G, et al. Among authors: negri l. J Med Chem. 2002 Dec 5;45(25):5556-63. doi: 10.1021/jm020336e. J Med Chem. 2002. PMID: 12459023

3

Synthesis and opioid activity of N,N-dimethyl-Dmt-Tic-NH-CH(R)-R' analogues: acquisition of potent delta antagonism.

Balboni G, Salvadori S, Guerrini R, Negri L, Giannini E, Bryant SD, Jinsmaa Y, Lazarus LH. Balboni G, et al. Among authors: negri l. Bioorg Med Chem. 2003 Dec 1;11(24):5435-41. doi: 10.1016/j.bmc.2003.09.039. Bioorg Med Chem. 2003. PMID: 14642588

4

Direct influence of C-terminally substituted amino acids in the Dmt-Tic pharmacophore on delta-opioid receptor selectivity and antagonism.

Balboni G, Salvadori S, Guerrini R, Negri L, Giannini E, Bryant SD, Jinsmaa Y, Lazarus LH. Balboni G, et al. Among authors: negri l. J Med Chem. 2004 Jul 29;47(16):4066-71. doi: 10.1021/jm040033f. J Med Chem. 2004. PMID: 15267245

5

Conversion of the potent delta-opioid agonist H-Dmt-Tic-NH-CH(2)-bid into delta-opioid antagonists by N(1)-benzimidazole alkylation(1).

Balboni G, Guerrini R, Salvadori S, Negri L, Giannini E, Bryant SD, Jinsmaa Y, Lazarus LH. Balboni G, et al. Among authors: negri l. J Med Chem. 2005 Dec 29;48(26):8112-4. doi: 10.1021/jm058259l. J Med Chem. 2005. PMID: 16366592 Free PMC article.

6

6-N,N-dimethylamino-2,3-naphthalimide: a new environment-sensitive fluorescent probe in delta- and mu-selective opioid peptides.

Vázquez ME, Blanco JB, Salvadori S, Trapella C, Argazzi R, Bryant SD, Jinsmaa Y, Lazarus LH, Negri L, Giannini E, Lattanzi R, Colucci M, Balboni G. Vázquez ME, et al. Among authors: negri l. J Med Chem. 2006 Jun 15;49(12):3653-8. doi: 10.1021/jm060343t. J Med Chem. 2006. PMID: 16759107 Free PMC article.

7

New 2',6'-dimethyl-L-tyrosine (Dmt) opioid peptidomimetics based on the Aba-Gly scaffold. Development of unique mu-opioid receptor ligands.

Ballet S, Salvadori S, Trapella C, Bryant SD, Jinsmaa Y, Lazarus LH, Negri L, Giannini E, Lattanzi R, Tourwé D, Balboni G. Ballet S, et al. Among authors: negri l. J Med Chem. 2006 Jun 29;49(13):3990-3. doi: 10.1021/jm0603264. J Med Chem. 2006. PMID: 16789756 Free PMC article.

8

A new opioid designed multiple ligand derived from the micro opioid agonist endomorphin-2 and the delta opioid antagonist pharmacophore Dmt-Tic.

Salvadori S, Trapella C, Fiorini S, Negri L, Lattanzi R, Bryant SD, Jinsmaa Y, Lazarus LH, Balboni G. Salvadori S, et al. Among authors: negri l. Bioorg Med Chem. 2007 Nov 15;15(22):6876-81. doi: 10.1016/j.bmc.2007.08.047. Epub 2007 Aug 29. Bioorg Med Chem. 2007. PMID: 17851080 Free PMC article.

9

Conformationally constrained opioid ligands: the Dmt-Aba and Dmt-Aia versus Dmt-Tic scaffold.

Ballet S, Feytens D, Wachter RD, Vlaeminck MD, Marczak ED, Salvadori S, Graaf Cd, Rognan D, Negri L, Lattanzi R, Lazarus LH, Tourwé D, Balboni G. Ballet S, et al. Among authors: negri l. Bioorg Med Chem Lett. 2009 Jan 15;19(2):433-7. doi: 10.1016/j.bmcl.2008.11.051. Epub 2008 Nov 19. Bioorg Med Chem Lett. 2009. PMID: 19062273 Free PMC article.

10

Synthesis and biological evaluation of 14-alkoxymorphinans. 22.(1) Influence of the 14-alkoxy group and the substitution in position 5 in 14-alkoxymorphinan-6-ones on in vitro and in vivo activities.

Lattanzi R, Spetea M, Schüllner F, Rief SB, Krassnig R, Negri L, Schmidhammer H. Lattanzi R, et al. Among authors: negri l. J Med Chem. 2005 May 5;48(9):3372-8. doi: 10.1021/jm040894o. J Med Chem. 2005. PMID: 15857143

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