Patch RJ - Search Results

1

2-Hydroxy-4,6-diamino-[1,3,5]triazines: a novel class of VEGF-R2 (KDR) tyrosine kinase inhibitors.

Baindur N, Chadha N, Brandt BM, Asgari D, Patch RJ, Schalk-Hihi C, Carver TE, Petrounia IP, Baumann CA, Ott H, Manthey C, Springer BA, Player MR. Baindur N, et al. Among authors: patch rj. J Med Chem. 2005 Mar 24;48(6):1717-20. doi: 10.1021/jm049372z. J Med Chem. 2005. PMID: 15771417

2

Identification of 2-acylaminothiophene-3-carboxamides as potent inhibitors of FLT3.

Patch RJ, Baumann CA, Liu J, Gibbs AC, Ott H, Lattanze J, Player MR. Patch RJ, et al. Bioorg Med Chem Lett. 2006 Jun 15;16(12):3282-6. doi: 10.1016/j.bmcl.2006.03.032. Epub 2006 Mar 31. Bioorg Med Chem Lett. 2006. PMID: 16580199

3

Potent 2'-aminoanilide inhibitors of cFMS as potential anti-inflammatory agents.

Patch RJ, Brandt BM, Asgari D, Baindur N, Chadha NK, Georgiadis T, Cheung WS, Petrounia IP, Donatelli RR, Chaikin MA, Player MR. Patch RJ, et al. Bioorg Med Chem Lett. 2007 Nov 15;17(22):6070-4. doi: 10.1016/j.bmcl.2007.09.057. Epub 2007 Sep 19. Bioorg Med Chem Lett. 2007. PMID: 17904845

4

Synthesis and evaluation of novel 3,4,6-substituted 2-quinolones as FMS kinase inhibitors.

Wall MJ, Chen J, Meegalla S, Ballentine SK, Wilson KJ, DesJarlais RL, Schubert C, Chaikin MA, Crysler C, Petrounia IP, Donatelli RR, Yurkow EJ, Boczon L, Mazzulla M, Player MR, Patch RJ, Manthey CL, Molloy C, Tomczuk B, Illig CR. Wall MJ, et al. Among authors: patch rj. Bioorg Med Chem Lett. 2008 Mar 15;18(6):2097-102. doi: 10.1016/j.bmcl.2008.01.088. Epub 2008 Jan 30. Bioorg Med Chem Lett. 2008. PMID: 18289848

5

A tandem Heck-carbocyclization/Suzuki-coupling approach to the stereoselective syntheses of asymmetric 3,3-(diarylmethylene)indolinones.

Cheung WS, Patch RJ, Player MR. Cheung WS, et al. Among authors: patch rj. J Org Chem. 2005 Apr 29;70(9):3741-4. doi: 10.1021/jo050016d. J Org Chem. 2005. PMID: 15845020

6

Single-step syntheses of 2-amino-7-chlorothiazolo[5,4-d]pyrimidines: intermediates for bivalent thiazolopyrimidines.

Liu J, Patch RJ, Schubert C, Player MR. Liu J, et al. Among authors: patch rj. J Org Chem. 2005 Nov 25;70(24):10194-7. doi: 10.1021/jo0517702. J Org Chem. 2005. PMID: 16292872

7

Crystal structure of the tyrosine kinase domain of colony-stimulating factor-1 receptor (cFMS) in complex with two inhibitors.

Schubert C, Schalk-Hihi C, Struble GT, Ma HC, Petrounia IP, Brandt B, Deckman IC, Patch RJ, Player MR, Spurlino JC, Springer BA. Schubert C, et al. Among authors: patch rj. J Biol Chem. 2007 Feb 9;282(6):4094-101. doi: 10.1074/jbc.M608183200. Epub 2006 Nov 28. J Biol Chem. 2007. PMID: 17132624 Free article.

8

Identification of diaryl ether-based ligands for estrogen-related receptor α as potential antidiabetic agents.

Patch RJ, Searle LL, Kim AJ, De D, Zhu X, Askari HB, O'Neill JC, Abad MC, Rentzeperis D, Liu J, Kemmerer M, Lin L, Kasturi J, Geisler JG, Lenhard JM, Player MR, Gaul MD. Patch RJ, et al. J Med Chem. 2011 Feb 10;54(3):788-808. doi: 10.1021/jm101063h. Epub 2011 Jan 10. J Med Chem. 2011. PMID: 21218783

9

Discovery of novel potent imidazo[1,2-b]pyridazine PDE10a inhibitors.

Meegalla SK, Huang H, Illig CR, Parks DJ, Chen J, Lee YK, Wilson KJ, Patel SK, Cheung WS, Lu T, Kirchner T, Askari HB, Geisler J, Patch RJ, Gibbs AC, Rady B, Connelly M, Player MR. Meegalla SK, et al. Among authors: patch rj. Bioorg Med Chem Lett. 2016 Sep 1;26(17):4216-22. doi: 10.1016/j.bmcl.2016.07.054. Epub 2016 Jul 25. Bioorg Med Chem Lett. 2016. PMID: 27491708

10

Indazole-based ligands for estrogen-related receptor α as potential anti-diabetic agents.

Patch RJ, Huang H, Patel S, Cheung W, Xu G, Zhao BP, Beauchamp DA, Rentzeperis D, Geisler JG, Askari HB, Liu J, Kasturi J, Towers M, Gaul MD, Player MR. Patch RJ, et al. Eur J Med Chem. 2017 Sep 29;138:830-853. doi: 10.1016/j.ejmech.2017.07.015. Epub 2017 Jul 14. Eur J Med Chem. 2017. PMID: 28735214

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