Čapková K - Search Results

1

Synthesis and evaluation of library of betulin derivatives against the botulinum neurotoxin A protease.

Šilhár P, Alakurtti S, Čapková K, Xiaochuan F, Shoemaker CB, Yli-Kauhaluoma J, Janda KD. Šilhár P, et al. Among authors: capkova k. Bioorg Med Chem Lett. 2011 Apr 15;21(8):2229-31. doi: 10.1016/j.bmcl.2011.02.115. Epub 2011 Mar 4. Bioorg Med Chem Lett. 2011. PMID: 21421315 Free PMC article.

2

Synthesis and structure-activity relationships of second-generation hydroxamate botulinum neurotoxin A protease inhibitors.

Capková K, Yoneda Y, Dickerson TJ, Janda KD. Capková K, et al. Bioorg Med Chem Lett. 2007 Dec 1;17(23):6463-6. doi: 10.1016/j.bmcl.2007.09.103. Epub 2007 Oct 9. Bioorg Med Chem Lett. 2007. PMID: 17951059 Free PMC article.

3

Toward the discovery of potent inhibitors of botulinum neurotoxin A: development of a robust LC MS based assay operational from low to subnanomolar enzyme concentrations.

Capková K, Hixon MS, McAllister LA, Janda KD. Capková K, et al. Chem Commun (Camb). 2008 Aug 14;(30):3525-7. doi: 10.1039/b808305c. Epub 2008 Jul 3. Chem Commun (Camb). 2008. PMID: 18654701

4

Investigations into small molecule non-peptidic inhibitors of the botulinum neurotoxins.

Capková K, Salzameda NT, Janda KD. Capková K, et al. Toxicon. 2009 Oct;54(5):575-82. doi: 10.1016/j.toxicon.2009.03.016. Epub 2009 Mar 25. Toxicon. 2009. PMID: 19327377 Free PMC article. Review.

5

Benzylidene cyclopentenediones: First irreversible inhibitors against botulinum neurotoxin A's zinc endopeptidase.

Capková K, Hixon MS, Pellett S, Barbieri JT, Johnson EA, Janda KD. Capková K, et al. Bioorg Med Chem Lett. 2010 Jan 1;20(1):206-8. doi: 10.1016/j.bmcl.2009.10.129. Epub 2009 Oct 31. Bioorg Med Chem Lett. 2010. PMID: 19914829 Free PMC article.

6

Botulinum neurotoxin A protease: discovery of natural product exosite inhibitors.

Silhár P, Capková K, Salzameda NT, Barbieri JT, Hixon MS, Janda KD. Silhár P, et al. Among authors: capkova k. J Am Chem Soc. 2010 Mar 10;132(9):2868-9. doi: 10.1021/ja910761y. J Am Chem Soc. 2010. PMID: 20158239 Free PMC article.

7

Evaluation of adamantane hydroxamates as botulinum neurotoxin inhibitors: synthesis, crystallography, modeling, kinetic and cellular based studies.

Šilhár P, Silvaggi NR, Pellett S, Čapková K, Johnson EA, Allen KN, Janda KD. Šilhár P, et al. Among authors: capkova k. Bioorg Med Chem. 2013 Mar 1;21(5):1344-8. doi: 10.1016/j.bmc.2012.12.001. Epub 2012 Dec 20. Bioorg Med Chem. 2013. PMID: 23340139 Free PMC article.

8

A cell-penetrating peptidic GRP78 ligand for tumor cell-specific prodrug therapy.

Yoneda Y, Steiniger SC, Capková K, Mee JM, Liu Y, Kaufmann GF, Janda KD. Yoneda Y, et al. Among authors: capkova k. Bioorg Med Chem Lett. 2008 Mar 1;18(5):1632-6. doi: 10.1016/j.bmcl.2008.01.060. Epub 2008 Jan 19. Bioorg Med Chem Lett. 2008. PMID: 18243696 Free PMC article.

9

Tissue factor-activated coagulation cascade in the tumor microenvironment is critical for tumor progression and an effective target for therapy.

Liu Y, Jiang P, Capkova K, Xue D, Ye L, Sinha SC, Mackman N, Janda KD, Liu C. Liu Y, et al. Among authors: capkova k. Cancer Res. 2011 Oct 15;71(20):6492-502. doi: 10.1158/0008-5472.CAN-11-1145. Epub 2011 Aug 31. Cancer Res. 2011. PMID: 21880589

10

Effects of hydroxamate metalloendoprotease inhibitors on botulinum neurotoxin A poisoned mouse neuromuscular junctions.

Thyagarajan B, Potian JG, Garcia CC, Hognason K, Capková K, Moe ST, Jacobson AR, Janda KD, McArdle JJ. Thyagarajan B, et al. Among authors: capkova k. Neuropharmacology. 2010 Jun;58(8):1189-98. doi: 10.1016/j.neuropharm.2010.02.014. Epub 2010 Mar 6. Neuropharmacology. 2010. PMID: 20211192 Free PMC article.

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