Matasi JJ - Search Results

1

Synthesis and SAR development of novel P2X7 receptor antagonists for the treatment of pain: part 2.

Brumfield S, Matasi JJ, Tulshian D, Czarniecki M, Greenlee W, Garlisi C, Qiu H, Devito K, Chen SC, Sun Y, Bertorelli R, Ansell J, Geiss W, Le VD, Martin GS, Vellekoop SA, Haber J, Allard ML. Brumfield S, et al. Among authors: matasi jj. Bioorg Med Chem Lett. 2011 Dec 15;21(24):7287-90. doi: 10.1016/j.bmcl.2011.10.037. Epub 2011 Oct 21. Bioorg Med Chem Lett. 2011. PMID: 22078214

2

Structure-activity relationships of 2,4-diphenyl-1H-imidazole analogs as CB2 receptor agonists for the treatment of chronic pain.

Yang SW, Smotryski J, Matasi J, Ho G, Tulshian D, Greenlee WJ, Brusa R, Beltramo M, Cox K. Yang SW, et al. Bioorg Med Chem Lett. 2011 Jan 1;21(1):182-5. doi: 10.1016/j.bmcl.2010.11.044. Epub 2010 Nov 11. Bioorg Med Chem Lett. 2011. PMID: 21115245

3

Initial optimization and series evolution of diaminopyrimidine inhibitors of interleukin-1 receptor associated kinase 4.

Seganish WM, McElroy WT, Herr RJ, Brumfield S, Greenlee WJ, Harding J, Komanduri V, Matasi J, Prakash KC, Tulshian D, Yang J, Yet L, Devito K, Fossetta J, Garlisi CG, Lundell D, Niu X, Sondey C. Seganish WM, et al. Bioorg Med Chem Lett. 2015 Aug 15;25(16):3203-7. doi: 10.1016/j.bmcl.2015.05.097. Epub 2015 Jun 6. Bioorg Med Chem Lett. 2015. PMID: 26115573

4

The discovery and synthesis of novel adenosine receptor (A(2A)) antagonists.

Matasi JJ, Caldwell JP, Hao J, Neustadt B, Arik L, Foster CJ, Lachowicz J, Tulshian DB. Matasi JJ, et al. Bioorg Med Chem Lett. 2005 Mar 1;15(5):1333-6. doi: 10.1016/j.bmcl.2005.01.019. Bioorg Med Chem Lett. 2005. PMID: 15713381

5

2-(2-Furanyl)-7-phenyl[1,2,4]triazolo[1,5-c]pyrimidin-5-amine analogs: highly potent, orally active, adenosine A2A antagonists. Part 1.

Matasi JJ, Caldwell JP, Zhang H, Fawzi A, Cohen-Williams ME, Varty GB, Tulshian DB. Matasi JJ, et al. Bioorg Med Chem Lett. 2005 Aug 15;15(16):3670-4. doi: 10.1016/j.bmcl.2005.05.086. Bioorg Med Chem Lett. 2005. PMID: 15978806

6

2-(2-Furanyl)-7-phenyl[1,2,4]triazolo[1,5-c]pyrimidin-5-amine analogs as adenosine A2A antagonists: the successful reduction of hERG activity. Part 2.

Matasi JJ, Caldwell JP, Zhang H, Fawzi A, Higgins GA, Cohen-Williams ME, Varty GB, Tulshian DB. Matasi JJ, et al. Bioorg Med Chem Lett. 2005 Aug 15;15(16):3675-8. doi: 10.1016/j.bmcl.2005.05.043. Bioorg Med Chem Lett. 2005. PMID: 15982882

7

3H-[1,2,4]-Triazolo[5,1-i]purin-5-amine derivatives as adenosine A2A antagonists.

Silverman LS, Caldwell JP, Greenlee WJ, Kiselgof E, Matasi JJ, Tulshian DB, Arik L, Foster C, Bertorelli R, Monopoli A, Ongini E. Silverman LS, et al. Among authors: matasi jj. Bioorg Med Chem Lett. 2007 Mar 15;17(6):1659-62. doi: 10.1016/j.bmcl.2006.12.104. Epub 2007 Jan 8. Bioorg Med Chem Lett. 2007. PMID: 17234414

8

Synthesis and structure-activity relationships of N-substituted spiropiperidines as nociceptin receptor ligands.

Caldwell JP, Matasi JJ, Zhang H, Fawzi A, Tulshian DB. Caldwell JP, et al. Among authors: matasi jj. Bioorg Med Chem Lett. 2007 Apr 15;17(8):2281-4. doi: 10.1016/j.bmcl.2007.01.069. Epub 2007 Jan 27. Bioorg Med Chem Lett. 2007. PMID: 17289383

9

Synthesis and structure-activity relationships of N-substituted spiropiperidines as nociceptin receptor ligands: part 2.

Caldwell JP, Matasi JJ, Fernandez X, McLeod RL, Zhang H, Fawzi A, Tulshian DB. Caldwell JP, et al. Among authors: matasi jj. Bioorg Med Chem Lett. 2009 Feb 15;19(4):1164-7. doi: 10.1016/j.bmcl.2008.12.092. Epub 2008 Dec 29. Bioorg Med Chem Lett. 2009. PMID: 19147350

10

Synthesis and SAR development of novel P2X7 receptor antagonists for the treatment of pain: part 1.

Matasi JJ, Brumfield S, Tulshian D, Czarnecki M, Greenlee W, Garlisi CG, Qiu H, Devito K, Chen SC, Sun Y, Bertorelli R, Geiss W, Le VD, Martin GS, Vellekoop SA, Haber J, Allard ML. Matasi JJ, et al. Bioorg Med Chem Lett. 2011 Jun 15;21(12):3805-8. doi: 10.1016/j.bmcl.2011.04.034. Epub 2011 Apr 24. Bioorg Med Chem Lett. 2011. PMID: 21570840

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