Jimenez HN - Search Results

1

Structure-activity relationships for negative allosteric mGluR5 modulators.

Kaae BH, Harpsøe K, Kvist T, Mathiesen JM, Mølck C, Gloriam D, Jimenez HN, Uberti MA, Nielsen SM, Nielsen B, Bräuner-Osborne H, Sauerberg P, Clausen RP, Madsen U. Kaae BH, et al. Among authors: jimenez hn. ChemMedChem. 2012 Mar 5;7(3):440-51. doi: 10.1002/cmdc.201100578. Epub 2012 Jan 20. ChemMedChem. 2012. PMID: 22267204

2

Pharmacological characterization and modeling of the binding sites of novel 1,3-bis(pyridinylethynyl)benzenes as metabotropic glutamate receptor 5-selective negative allosteric modulators.

Mølck C, Harpsøe K, Gloriam DE, Clausen RP, Madsen U, Pedersen LØ, Jimenez HN, Nielsen SM, Mathiesen JM, Bräuner-Osborne H. Mølck C, et al. Among authors: jimenez hn. Mol Pharmacol. 2012 Nov;82(5):929-37. doi: 10.1124/mol.112.078808. Epub 2012 Aug 16. Mol Pharmacol. 2012. PMID: 22899869

3

6-Aryl-3-pyrrolidinylpyridines as mGlu5 receptor negative allosteric modulators.

Weiss JM, Jimenez HN, Li G, April M, Uberti MA, Bacolod MD, Brodbeck RM, Doller D. Weiss JM, et al. Among authors: jimenez hn. Bioorg Med Chem Lett. 2011 Aug 15;21(16):4891-9. doi: 10.1016/j.bmcl.2011.06.014. Epub 2011 Jun 17. Bioorg Med Chem Lett. 2011. PMID: 21757343

4

4-(1-Phenyl-1H-pyrazol-4-yl)quinolines as novel, selective and brain penetrant metabotropic glutamate receptor 4 positive allosteric modulators.

Jimenez HN, Liu KG, Hong SP, Reitman MS, Uberti MA, Bacolod MD, Cajina M, Nattini M, Sabio M, Doller D. Jimenez HN, et al. Bioorg Med Chem Lett. 2012 May 1;22(9):3235-9. doi: 10.1016/j.bmcl.2012.03.032. Epub 2012 Mar 15. Bioorg Med Chem Lett. 2012. PMID: 22465637

5

Discovery and structure-activity relationship of 1,3-cyclohexyl amide derivatives as novel mGluR5 negative allosteric modulators.

Zhou H, Topiol SW, Grenon M, Jimenez HN, Uberti MA, Smith DG, Brodbeck RM, Chandrasena G, Pedersen H, Madsen JC, Doller D, Li G. Zhou H, et al. Among authors: jimenez hn. Bioorg Med Chem Lett. 2013 Mar 1;23(5):1398-406. doi: 10.1016/j.bmcl.2012.12.078. Epub 2013 Jan 5. Bioorg Med Chem Lett. 2013. PMID: 23357634

6

Synergy between L-DOPA and a novel positive allosteric modulator of metabotropic glutamate receptor 4: implications for Parkinson's disease treatment and dyskinesia.

Bennouar KE, Uberti MA, Melon C, Bacolod MD, Jimenez HN, Cajina M, Kerkerian-Le Goff L, Doller D, Gubellini P. Bennouar KE, et al. Among authors: jimenez hn. Neuropharmacology. 2013 Mar;66:158-69. doi: 10.1016/j.neuropharm.2012.03.022. Epub 2012 Apr 3. Neuropharmacology. 2013. PMID: 22491024

7

5-(2'-Pyridyl)-2-aminothiazoles: alkyl amino sulfonamides and sulfamides as potent NPY(5) antagonists.

Packiarajan M, Coate H, Desai M, Jimenez HN, Reinhard EJ, Jubian VJ, Marzabadi MR, Chandrasena G, Wolinski TC, Walker MW, Andersen K. Packiarajan M, et al. Among authors: jimenez hn. Bioorg Med Chem Lett. 2011 Nov 1;21(21):6500-4. doi: 10.1016/j.bmcl.2011.08.072. Epub 2011 Aug 28. Bioorg Med Chem Lett. 2011. PMID: 21924902

8

Amino substituted analogs of 1-phenyl-3-phenylimino-2-indolones with potent galanin Gal3 receptor binding affinity and improved solubility.

Konkel MJ, Packiarajan M, Chen H, Topiwala UP, Jimenez H, Talisman IJ, Coate H, Walker MW. Konkel MJ, et al. Bioorg Med Chem Lett. 2006 Aug 1;16(15):3950-4. doi: 10.1016/j.bmcl.2006.05.025. Epub 2006 May 30. Bioorg Med Chem Lett. 2006. PMID: 16730981

9

3-arylimino-2-indolones are potent and selective galanin GAL3 receptor antagonists.

Konkel MJ, Lagu B, Boteju LW, Jimenez H, Noble S, Walker MW, Chandrasena G, Blackburn TP, Nikam SS, Wright JL, Kornberg BE, Gregory T, Pugsley TA, Akunne H, Zoski K, Wise LD. Konkel MJ, et al. J Med Chem. 2006 Jun 29;49(13):3757-8. doi: 10.1021/jm060001n. J Med Chem. 2006. PMID: 16789730

10

Novel bioactive and stable neurotensin peptide analogues capable of delivering radiopharmaceuticals and molecular beacons to tumors.

Achilefu S, Srinivasan A, Schmidt MA, Jimenez HN, Bugaj JE, Erion JL. Achilefu S, et al. Among authors: jimenez hn. J Med Chem. 2003 Jul 17;46(15):3403-11. doi: 10.1021/jm030081k. J Med Chem. 2003. PMID: 12852770

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