Pin JP - Search Results

1

OptoGluNAM4.1, a Photoswitchable Allosteric Antagonist for Real-Time Control of mGlu4 Receptor Activity.

Rovira X, Trapero A, Pittolo S, Zussy C, Faucherre A, Jopling C, Giraldo J, Pin JP, Gorostiza P, Goudet C, Llebaria A. Rovira X, et al. Among authors: pin jp. Cell Chem Biol. 2016 Aug 18;23(8):929-34. doi: 10.1016/j.chembiol.2016.06.013. Epub 2016 Jul 28. Cell Chem Biol. 2016. PMID: 27478159 Free article.

2

Heptahelical domain of metabotropic glutamate receptor 5 behaves like rhodopsin-like receptors.

Goudet C, Gaven F, Kniazeff J, Vol C, Liu J, Cohen-Gonsaud M, Acher F, Prézeau L, Pin JP. Goudet C, et al. Among authors: pin jp. Proc Natl Acad Sci U S A. 2004 Jan 6;101(1):378-83. doi: 10.1073/pnas.0304699101. Epub 2003 Dec 22. Proc Natl Acad Sci U S A. 2004. PMID: 14691258 Free PMC article.

3

Locking the dimeric GABA(B) G-protein-coupled receptor in its active state.

Kniazeff J, Saintot PP, Goudet C, Liu J, Charnet A, Guillon G, Pin JP. Kniazeff J, et al. Among authors: pin jp. J Neurosci. 2004 Jan 14;24(2):370-7. doi: 10.1523/JNEUROSCI.3141-03.2004. J Neurosci. 2004. PMID: 14724235 Free PMC article.

4

Evidence for a single heptahelical domain being turned on upon activation of a dimeric GPCR.

Hlavackova V, Goudet C, Kniazeff J, Zikova A, Maurel D, Vol C, Trojanova J, Prézeau L, Pin JP, Blahos J. Hlavackova V, et al. Among authors: pin jp. EMBO J. 2005 Feb 9;24(3):499-509. doi: 10.1038/sj.emboj.7600557. Epub 2005 Jan 20. EMBO J. 2005. PMID: 15660124 Free PMC article.

5

Asymmetric functioning of dimeric metabotropic glutamate receptors disclosed by positive allosteric modulators.

Goudet C, Kniazeff J, Hlavackova V, Malhaire F, Maurel D, Acher F, Blahos J, Prézeau L, Pin JP. Goudet C, et al. Among authors: pin jp. J Biol Chem. 2005 Jul 1;280(26):24380-5. doi: 10.1074/jbc.M502642200. Epub 2005 Apr 29. J Biol Chem. 2005. PMID: 15863499 Free PMC article.

6

Interaction of novel positive allosteric modulators of metabotropic glutamate receptor 5 with the negative allosteric antagonist site is required for potentiation of receptor responses.

Chen Y, Nong Y, Goudet C, Hemstapat K, de Paulis T, Pin JP, Conn PJ. Chen Y, et al. Among authors: pin jp. Mol Pharmacol. 2007 May;71(5):1389-98. doi: 10.1124/mol.106.032425. Epub 2007 Feb 15. Mol Pharmacol. 2007. PMID: 17303702

7

Synthesis and biological evaluation of 1-amino-2-phosphonomethylcyclopropanecarboxylic acids, new group III metabotropic glutamate receptor agonists.

Sibille P, Lopez S, Brabet I, Valenti O, Oueslati N, Gaven F, Goudet C, Bertrand HO, Neyton J, Marino MJ, Amalric M, Pin JP, Acher FC. Sibille P, et al. Among authors: pin jp. J Med Chem. 2007 Jul 26;50(15):3585-95. doi: 10.1021/jm070262c. Epub 2007 Jun 28. J Med Chem. 2007. PMID: 17602546

8

L-(+)-2-Amino-4-thiophosphonobutyric acid (L-thioAP4), a new potent agonist of group III metabotropic glutamate receptors: increased distal acidity affords enhanced potency.

Selvam C, Goudet C, Oueslati N, Pin JP, Acher FC. Selvam C, et al. Among authors: pin jp. J Med Chem. 2007 Sep 20;50(19):4656-64. doi: 10.1021/jm070400y. Epub 2007 Aug 28. J Med Chem. 2007. PMID: 17722902

9

Group III metabotropic glutamate receptors inhibit hyperalgesia in animal models of inflammation and neuropathic pain.

Goudet C, Chapuy E, Alloui A, Acher F, Pin JP, Eschalier A. Goudet C, et al. Among authors: pin jp. Pain. 2008 Jul;137(1):112-124. doi: 10.1016/j.pain.2007.08.020. Epub 2007 Sep 27. Pain. 2008. PMID: 17900808 Free article.

10

N-{4-Chloro-2-[(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)methyl]phenyl}-2-hydroxybenzamide (CPPHA) acts through a novel site as a positive allosteric modulator of group 1 metabotropic glutamate receptors.

Chen Y, Goudet C, Pin JP, Conn PJ. Chen Y, et al. Among authors: pin jp. Mol Pharmacol. 2008 Mar;73(3):909-18. doi: 10.1124/mol.107.040097. Epub 2007 Dec 4. Mol Pharmacol. 2008. PMID: 18056795

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