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Page 1
Identification of (R)-N-((4-Methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methyl-1-(1-(1-(2,2,2-trifluoroethyl)piperidin-4-yl)ethyl)-1H-indole-3-carboxamide (CPI-1205), a Potent and Selective Inhibitor of Histone Methyltransferase EZH2, Suitable for Phase I Clinical Trials for B-Cell Lymphomas.
Vaswani RG, Gehling VS, Dakin LA, Cook AS, Nasveschuk CG, Duplessis M, Iyer P, Balasubramanian S, Zhao F, Good AC, Campbell R, Lee C, Cantone N, Cummings RT, Normant E, Bellon SF, Albrecht BK, Harmange JC, Trojer P, Audia JE, Zhang Y, Justin N, Chen S, Wilson JR, Gamblin SJ. Vaswani RG, et al. Among authors: iyer p. J Med Chem. 2016 Nov 10;59(21):9928-9941. doi: 10.1021/acs.jmedchem.6b01315. Epub 2016 Oct 28. J Med Chem. 2016. PMID: 27739677 Free PMC article.
Discovery, design, and synthesis of indole-based EZH2 inhibitors.
Gehling VS, Vaswani RG, Nasveschuk CG, Duplessis M, Iyer P, Balasubramanian S, Zhao F, Good AC, Campbell R, Lee C, Dakin LA, Cook AS, Gagnon A, Harmange JC, Audia JE, Cummings RT, Normant E, Trojer P, Albrecht BK. Gehling VS, et al. Among authors: iyer p. Bioorg Med Chem Lett. 2015 Sep 1;25(17):3644-9. doi: 10.1016/j.bmcl.2015.06.056. Epub 2015 Jun 19. Bioorg Med Chem Lett. 2015. PMID: 26189078
Design and Synthesis of Styrenylcyclopropylamine LSD1 Inhibitors.
Gehling VS, McGrath JP, Duplessis M, Khanna A, Brucelle F, Vaswani RG, Côté A, Stuckey J, Watson V, Cummings RT, Balasubramanian S, Iyer P, Sawant P, Good AC, Albrecht BK, Harmange JC, Audia JE, Bellon SF, Trojer P, Levell JR. Gehling VS, et al. Among authors: iyer p. ACS Med Chem Lett. 2020 May 6;11(6):1213-1220. doi: 10.1021/acsmedchemlett.0c00060. eCollection 2020 Jun 11. ACS Med Chem Lett. 2020. PMID: 32551003 Free PMC article.
EZH2 inhibitor efficacy in non-Hodgkin's lymphoma does not require suppression of H3K27 monomethylation.
Bradley WD, Arora S, Busby J, Balasubramanian S, Gehling VS, Nasveschuk CG, Vaswani RG, Yuan CC, Hatton C, Zhao F, Williamson KE, Iyer P, Méndez J, Campbell R, Cantone N, Garapaty-Rao S, Audia JE, Cook AS, Dakin LA, Albrecht BK, Harmange JC, Daniels DL, Cummings RT, Bryant BM, Normant E, Trojer P. Bradley WD, et al. Among authors: iyer p. Chem Biol. 2014 Nov 20;21(11):1463-75. doi: 10.1016/j.chembiol.2014.09.017. Chem Biol. 2014. PMID: 25457180
Quality indicators for upper GI endoscopy.
Yadlapati R, Early D, Iyer PG, Morgan DR, Sengupta N, Sharma P, Shaheen NJ. Yadlapati R, et al. Among authors: iyer pg. Gastrointest Endosc. 2024 Nov 13:S0016-5107(24)03460-6. doi: 10.1016/j.gie.2024.08.023. Online ahead of print. Gastrointest Endosc. 2024. PMID: 39545899 No abstract available.
Patterns of loco-regional progression and patient outcomes after definitive-dose radiation therapy for anaplastic thyroid cancer.
Bronk JK, Augustyn A, Mohamed ASR, David Fuller C, Garden AS, Moreno AC, Lee A, Morrison WH, Phan J, Reddy JP, Rosenthal DI, Spiotto MT, Frank SJ, Dadu R, Busaidy N, Zafereo M, Wang JR, Maniakas A, Ferrarotto R, Iyer PC, Cabanillas ME, Gunn GB. Bronk JK, et al. Among authors: iyer pc. Radiother Oncol. 2024 Nov 1;202:110602. doi: 10.1016/j.radonc.2024.110602. Online ahead of print. Radiother Oncol. 2024. PMID: 39489425 Free article.
Roadmap on magnetic nanoparticles in nanomedicine.
Wu K, Wang JP, Natekar NA, Ciannella S, González-Fernández C, Gomez-Pastora J, Bao Y, Liu J, Liang S, Wu X, Nguyen T Tran L, Mercedes Paz González K, Choe H, Strayer J, Iyer PR, Chalmers J, Chugh VK, Rezaei B, Mostufa S, Tay ZW, Saayujya C, Huynh Q, Bryan J, Kuo R, Yu E, Chandrasekharan P, Fellows B, Conolly S, Hadimani RL, El-Gendy AA, Saha R, Broomhall TJ, Wright AL, Rotherham M, El Haj AJ, Wang Z, Liang J, Abad-Díaz-de-Cerio A, Gandarias L, Gubieda AG, García-Prieto A, Fdez-Gubieda ML. Wu K, et al. Among authors: iyer pr. Nanotechnology. 2024 Nov 5;36(4):042003. doi: 10.1088/1361-6528/ad8626. Nanotechnology. 2024. PMID: 39395441 Free PMC article. Review.
920 results