Yan G - Search Results

1

Design, Synthesis, and Biological Evaluation of Dimorpholine Substituted Thienopyrimidines as Potential Class I PI3K/mTOR Dual Inhibitors.

Zhan M, Deng Y, Zhao L, Yan G, Wang F, Tian Y, Zhang L, Jiang H, Chen Y. Zhan M, et al. Among authors: yan g. J Med Chem. 2017 May 11;60(9):4023-4035. doi: 10.1021/acs.jmedchem.7b00357. Epub 2017 Apr 24. J Med Chem. 2017. PMID: 28409639

2

Synthesis and biological evaluation of 4-(1,2,3-triazol-1-yl)coumarin derivatives as potential antitumor agents.

Zhang W, Li Z, Zhou M, Wu F, Hou X, Luo H, Liu H, Han X, Yan G, Ding Z, Li R. Zhang W, et al. Among authors: yan g. Bioorg Med Chem Lett. 2014 Feb 1;24(3):799-807. doi: 10.1016/j.bmcl.2013.12.095. Epub 2013 Dec 29. Bioorg Med Chem Lett. 2014. PMID: 24418772

3

Synthesis and biological evaluation of novel 2,3-dihydrochromeno[3,4-d]imidazol-4(1H)-one derivatives as potent anticancer cell proliferation and migration agents.

Han X, Luo J, Wu F, Hou X, Yan G, Zhou M, Zhang M, Pu C, Li R. Han X, et al. Among authors: yan g. Eur J Med Chem. 2016 May 23;114:232-43. doi: 10.1016/j.ejmech.2016.01.035. Epub 2016 Feb 5. Eur J Med Chem. 2016. PMID: 26994691

4

Synthesis, biological evaluation and molecular docking study of N-(2-methoxyphenyl)-6-((4-nitrophenyl)sulfonyl)benzamide derivatives as potent HIV-1 Vif antagonists.

Zhou M, Luo RH, Hou XY, Wang RR, Yan GY, Chen H, Zhang RH, Shi JY, Zheng YT, Li R, Wei YQ. Zhou M, et al. Eur J Med Chem. 2017 Mar 31;129:310-324. doi: 10.1016/j.ejmech.2017.01.010. Epub 2017 Jan 12. Eur J Med Chem. 2017. PMID: 28235704

5

Design, synthesis and biological evaluation of indole derivatives as Vif inhibitors.

Pu C, Luo RH, Zhang M, Hou X, Yan G, Luo J, Zheng YT, Li R. Pu C, et al. Among authors: yan g. Bioorg Med Chem Lett. 2017 Sep 1;27(17):4150-4155. doi: 10.1016/j.bmcl.2017.07.026. Epub 2017 Jul 10. Bioorg Med Chem Lett. 2017. PMID: 28754362

6

Discovery of a novel class of pyridine derivatives that selectively inhibits mutant isocitrate dehydrogenase 2.

Wang F, Li Z, Zhang T, Yan G, Hu M, Zhao L, Zhao Y, Chen Y. Wang F, et al. Among authors: yan g. Chem Biol Drug Des. 2018 Jun;91(6):1087-1093. doi: 10.1111/cbdd.13139. Epub 2018 Mar 30. Chem Biol Drug Des. 2018. PMID: 29120536

7

Discovery and biological evaluation of novel androgen receptor antagonist for castration-resistant prostate cancer.

Yu J, Zhang L, Yan G, Zhou P, Cao C, Zhou F, Li X, Chen Y. Yu J, et al. Among authors: yan g. Eur J Med Chem. 2019 Jun 1;171:265-281. doi: 10.1016/j.ejmech.2019.03.041. Epub 2019 Mar 22. Eur J Med Chem. 2019. PMID: 30925341

8

Discovery of 4-phenyl-2H-benzo[b][1,4]oxazin-3(4H)-one derivatives as potent and orally active PI3K/mTOR dual inhibitors.

Yan G, Pu C, Lan S, Zhong X, Zhou M, Hou X, Yang J, Shan H, Zhao L, Li R. Yan G, et al. Eur J Med Chem. 2019 Sep 15;178:667-686. doi: 10.1016/j.ejmech.2019.06.021. Epub 2019 Jun 13. Eur J Med Chem. 2019. PMID: 31228810

9

Discovery and biological evaluation of darolutamide derivatives as inhibitors and down-regulators of wild-type AR and the mutants.

Yu J, Zhou P, Hu M, Yang L, Yan G, Xu R, Deng Y, Li X, Chen Y. Yu J, et al. Among authors: yan g. Eur J Med Chem. 2019 Nov 15;182:111608. doi: 10.1016/j.ejmech.2019.111608. Epub 2019 Aug 10. Eur J Med Chem. 2019. PMID: 31437779

10

Design, synthesis, and biological evaluation of 2-amino-N-(2-methoxyphenyl)-6-((4-nitrophenyl)sulfonyl)benzamide derivatives as potent HIV-1 Vif inhibitors.

Zhang RH, Wang S, Luo RH, Zhou M, Zhang H, Xu GB, Zhao YL, Li YJ, Wang YL, Yan G, Liao SG, Zheng YT, Li R. Zhang RH, et al. Among authors: yan g. Bioorg Med Chem Lett. 2019 Dec 15;29(24):126638. doi: 10.1016/j.bmcl.2019.126638. Epub 2019 Aug 28. Bioorg Med Chem Lett. 2019. PMID: 31685340

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