Ding K - Search Results

1

Inhibition of Discoidin Domain Receptor 1 Reduces Collagen-mediated Tumorigenicity in Pancreatic Ductal Adenocarcinoma.

Aguilera KY, Huang H, Du W, Hagopian MM, Wang Z, Hinz S, Hwang TH, Wang H, Fleming JB, Castrillon DH, Ren X, Ding K, Brekken RA. Aguilera KY, et al. Among authors: ding k. Mol Cancer Ther. 2017 Nov;16(11):2473-2485. doi: 10.1158/1535-7163.MCT-16-0834. Epub 2017 Sep 1. Mol Cancer Ther. 2017. PMID: 28864681 Free PMC article.

2

A new diaryl urea compound, D181, induces cell cycle arrest in the G1 and M phases by targeting receptor tyrosine kinases and the microtubule skeleton.

Zhang J, Zhou J, Ren X, Diao Y, Li H, Jiang H, Ding K, Pei D. Zhang J, et al. Among authors: ding k. Invest New Drugs. 2012 Apr;30(2):490-507. doi: 10.1007/s10637-010-9577-1. Epub 2010 Nov 16. Invest New Drugs. 2012. PMID: 21080210

3

Identification of pyrido[1,2-α]pyrimidine-4-ones as new molecules improving the transcriptional functions of estrogen-related receptor α.

Peng L, Gao X, Duan L, Ren X, Wu D, Ding K. Peng L, et al. Among authors: ding k. J Med Chem. 2011 Nov 10;54(21):7729-33. doi: 10.1021/jm200976s. Epub 2011 Oct 12. J Med Chem. 2011. PMID: 21958216

4

Design, synthesis, and biological evaluation of novel conformationally constrained inhibitors targeting epidermal growth factor receptor threonine⁷⁹⁰ → methionine⁷⁹⁰ mutant.

Chang S, Zhang L, Xu S, Luo J, Lu X, Zhang Z, Xu T, Liu Y, Tu Z, Xu Y, Ren X, Geng M, Ding J, Pei D, Ding K. Chang S, et al. Among authors: ding k, ding j. J Med Chem. 2012 Mar 22;55(6):2711-23. doi: 10.1021/jm201591k. Epub 2012 Mar 1. J Med Chem. 2012. PMID: 22339342

5

Discovery and optimization of 3-(2-(Pyrazolo[1,5-a]pyrimidin-6-yl)ethynyl)benzamides as novel selective and orally bioavailable discoidin domain receptor 1 (DDR1) inhibitors.

Gao M, Duan L, Luo J, Zhang L, Lu X, Zhang Y, Zhang Z, Tu Z, Xu Y, Ren X, Ding K. Gao M, et al. Among authors: ding k. J Med Chem. 2013 Apr 25;56(8):3281-95. doi: 10.1021/jm301824k. Epub 2013 Apr 10. J Med Chem. 2013. PMID: 23521020

6

1-Phenyl-4-benzoyl-1H-1,2,3-triazoles as orally bioavailable transcriptional function suppressors of estrogen-related receptor α.

Xu S, Zhuang X, Pan X, Zhang Z, Duan L, Liu Y, Zhang L, Ren X, Ding K. Xu S, et al. Among authors: ding k. J Med Chem. 2013 Jun 13;56(11):4631-40. doi: 10.1021/jm4003928. Epub 2013 May 24. J Med Chem. 2013. PMID: 23656512

7

Pyrimido[4,5-d]pyrimidin-4(1H)-one derivatives as selective inhibitors of EGFR threonine790 to methionine790 (T790M) mutants.

Xu T, Zhang L, Xu S, Yang CY, Luo J, Ding F, Lu X, Liu Y, Tu Z, Li S, Pei D, Cai Q, Li H, Ren X, Wang S, Ding K. Xu T, et al. Among authors: ding k, ding f. Angew Chem Int Ed Engl. 2013 Aug 5;52(32):8387-90. doi: 10.1002/anie.201302313. Epub 2013 Jun 26. Angew Chem Int Ed Engl. 2013. PMID: 23804305 Free article. No abstract available.

8

Design, synthesis, and biological evaluation of 2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidinyl derivatives as new irreversible epidermal growth factor receptor inhibitors with improved pharmacokinetic properties.

Xu S, Xu T, Zhang L, Zhang Z, Luo J, Liu Y, Lu X, Tu Z, Ren X, Ding K. Xu S, et al. Among authors: ding k. J Med Chem. 2013 Nov 14;56(21):8803-13. doi: 10.1021/jm4012388. Epub 2013 Oct 31. J Med Chem. 2013. PMID: 24124898

9

Identification and optimization of new dual inhibitors of B-Raf and epidermal growth factor receptor kinases for overcoming resistance against vemurafenib.

Cheng H, Chang Y, Zhang L, Luo J, Tu Z, Lu X, Zhang Q, Lu J, Ren X, Ding K. Cheng H, et al. Among authors: ding k. J Med Chem. 2014 Mar 27;57(6):2692-703. doi: 10.1021/jm500007h. Epub 2014 Mar 18. J Med Chem. 2014. PMID: 24588073

10

Antitumor activity of S116836, a novel tyrosine kinase inhibitor, against imatinib-resistant FIP1L1-PDGFRα-expressing cells.

Shen Y, Ren X, Ding K, Zhang Z, Wang D, Pan J. Shen Y, et al. Among authors: ding k. Oncotarget. 2014 Nov 15;5(21):10407-20. doi: 10.18632/oncotarget.2090. Oncotarget. 2014. PMID: 25431951 Free PMC article.

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