Evers A - Search Results

1

Peptide Optimization at the Drug Discovery-Development Interface: Tailoring of Physicochemical Properties Toward Specific Formulation Requirements.

Evers A, Pfeiffer-Marek S, Bossart M, Heubel C, Stock U, Tiwari G, Gebauer B, Elshorst B, Pfenninger A, Lukasczyk U, Hessler G, Kamm W, Wagner M. Evers A, et al. J Pharm Sci. 2019 Apr;108(4):1404-1414. doi: 10.1016/j.xphs.2018.11.043. Epub 2018 Dec 4. J Pharm Sci. 2019. PMID: 30528197

2

Virtual screening of biogenic amine-binding G-protein coupled receptors: comparative evaluation of protein- and ligand-based virtual screening protocols.

Evers A, Hessler G, Matter H, Klabunde T. Evers A, et al. J Med Chem. 2005 Aug 25;48(17):5448-65. doi: 10.1021/jm050090o. J Med Chem. 2005. PMID: 16107144

3

Multiple-ligand-based virtual screening: methods and applications of the MTree approach.

Hessler G, Zimmermann M, Matter H, Evers A, Naumann T, Lengauer T, Rarey M. Hessler G, et al. Among authors: evers a. J Med Chem. 2005 Oct 20;48(21):6575-84. doi: 10.1021/jm050078w. J Med Chem. 2005. PMID: 16220974

4

Identification of high-affinity P2Y₁₂ antagonists based on a phenylpyrazole glutamic acid piperazine backbone.

Zech G, Hessler G, Evers A, Weiss T, Florian P, Just M, Czech J, Czechtizky W, Görlitzer J, Ruf S, Kohlmann M, Nazaré M. Zech G, et al. Among authors: evers a. J Med Chem. 2012 Oct 25;55(20):8615-29. doi: 10.1021/jm300771j. Epub 2012 Oct 4. J Med Chem. 2012. PMID: 22984835

5

CROSS: an efficient workflow for reaction-driven rescaffolding and side-chain optimization using robust chemical reactions and available reagents.

Evers A, Hessler G, Wang LH, Werrel S, Monecke P, Matter H. Evers A, et al. J Med Chem. 2013 Jun 13;56(11):4656-70. doi: 10.1021/jm400404v. Epub 2013 May 16. J Med Chem. 2013. PMID: 23627295

6

Recent progress and future options in the development of GLP-1 receptor agonists for the treatment of diabesity.

Lorenz M, Evers A, Wagner M. Lorenz M, et al. Among authors: evers a. Bioorg Med Chem Lett. 2013 Jul 15;23(14):4011-8. doi: 10.1016/j.bmcl.2013.05.022. Epub 2013 May 16. Bioorg Med Chem Lett. 2013. PMID: 23743288 Free article. Review.

7

Design of Novel Exendin-Based Dual Glucagon-like Peptide 1 (GLP-1)/Glucagon Receptor Agonists.

Evers A, Haack T, Lorenz M, Bossart M, Elvert R, Henkel B, Stengelin S, Kurz M, Glien M, Dudda A, Lorenz K, Kadereit D, Wagner M. Evers A, et al. J Med Chem. 2017 May 25;60(10):4293-4303. doi: 10.1021/acs.jmedchem.7b00174. Epub 2017 May 5. J Med Chem. 2017. PMID: 28448133

8

Dual Glucagon-like Peptide 1 (GLP-1)/Glucagon Receptor Agonists Specifically Optimized for Multidose Formulations.

Evers A, Bossart M, Pfeiffer-Marek S, Elvert R, Schreuder H, Kurz M, Stengelin S, Lorenz M, Herling A, Konkar A, Lukasczyk U, Pfenninger A, Lorenz K, Haack T, Kadereit D, Wagner M. Evers A, et al. J Med Chem. 2018 Jul 12;61(13):5580-5593. doi: 10.1021/acs.jmedchem.8b00292. Epub 2018 Jun 25. J Med Chem. 2018. PMID: 29879354

9

Running on mixed fuel-dual agonistic approach of GLP-1 and GCG receptors leads to beneficial impact on body weight and blood glucose control: A comparative study between mice and non-human primates.

Elvert R, Herling AW, Bossart M, Weiss T, Zhang B, Wenski P, Wandschneider J, Kleutsch S, Butty U, Kannt A, Wagner M, Haack T, Evers A, Dudda A, Lorenz M, Keil S, Larsen PJ. Elvert R, et al. Among authors: evers a. Diabetes Obes Metab. 2018 Aug;20(8):1836-1851. doi: 10.1111/dom.13212. Epub 2018 Jun 25. Diabetes Obes Metab. 2018. PMID: 29938884 Free PMC article.

10

Team Players or Opponents: Coadministration of Selective Glucagon and GLP-1 Receptor Agonists in Obese Diabetic Monkeys.

Elvert R, Bossart M, Herling AW, Weiss T, Zhang B, Kannt A, Wagner M, Haack T, Evers A, Dudda A, Keil S, Lorenz M, Lorenz K, Riz M, Hennerici W, Larsen PJ. Elvert R, et al. Among authors: evers a. Endocrinology. 2018 Aug 1;159(8):3105-3119. doi: 10.1210/en.2018-00399. Endocrinology. 2018. PMID: 29992313

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