Bräuner-Osborne H - Search Results

1

Identification of a novel scaffold for a small molecule GPR139 receptor agonist.

Nøhr AC, Shehata MA, Palmer D, Pokhrel R, Vallianou M, Foster SR, Gentry PR, Gloriam DE, Bräuner-Osborne H. Nøhr AC, et al. Sci Rep. 2019 Mar 7;9(1):3802. doi: 10.1038/s41598-019-40085-9. Sci Rep. 2019. PMID: 30846711 Free PMC article.

2

Chemogenomic discovery of allosteric antagonists at the GPRC6A receptor.

Gloriam DE, Wellendorph P, Johansen LD, Thomsen AR, Phonekeo K, Pedersen DS, Bräuner-Osborne H. Gloriam DE, et al. Chem Biol. 2011 Nov 23;18(11):1489-98. doi: 10.1016/j.chembiol.2011.09.012. Chem Biol. 2011. PMID: 22118683

3

Structure-activity relationships for negative allosteric mGluR5 modulators.

Kaae BH, Harpsøe K, Kvist T, Mathiesen JM, Mølck C, Gloriam D, Jimenez HN, Uberti MA, Nielsen SM, Nielsen B, Bräuner-Osborne H, Sauerberg P, Clausen RP, Madsen U. Kaae BH, et al. ChemMedChem. 2012 Mar 5;7(3):440-51. doi: 10.1002/cmdc.201100578. Epub 2012 Jan 20. ChemMedChem. 2012. PMID: 22267204

4

Pharmacological characterization and modeling of the binding sites of novel 1,3-bis(pyridinylethynyl)benzenes as metabotropic glutamate receptor 5-selective negative allosteric modulators.

Mølck C, Harpsøe K, Gloriam DE, Clausen RP, Madsen U, Pedersen LØ, Jimenez HN, Nielsen SM, Mathiesen JM, Bräuner-Osborne H. Mølck C, et al. Mol Pharmacol. 2012 Nov;82(5):929-37. doi: 10.1124/mol.112.078808. Epub 2012 Aug 16. Mol Pharmacol. 2012. PMID: 22899869

5

The GPCR, class C, group 6, subtype A (GPRC6A) receptor: from cloning to physiological function.

Clemmensen C, Smajilovic S, Wellendorph P, Bräuner-Osborne H. Clemmensen C, et al. Br J Pharmacol. 2014 Mar;171(5):1129-41. doi: 10.1111/bph.12365. Br J Pharmacol. 2014. PMID: 24032653 Free PMC article. Review.

6

Crystal structure and pharmacological characterization of a novel N-methyl-D-aspartate (NMDA) receptor antagonist at the GluN1 glycine binding site.

Kvist T, Steffensen TB, Greenwood JR, Mehrzad Tabrizi F, Hansen KB, Gajhede M, Pickering DS, Traynelis SF, Kastrup JS, Bräuner-Osborne H. Kvist T, et al. J Biol Chem. 2013 Nov 15;288(46):33124-35. doi: 10.1074/jbc.M113.480210. Epub 2013 Sep 26. J Biol Chem. 2013. PMID: 24072709 Free PMC article.

7

mGluR5: exploration of orthosteric and allosteric ligand binding pockets and their applications to drug discovery.

Mølck C, Harpsøe K, Gloriam DE, Mathiesen JM, Nielsen SM, Bräuner-Osborne H. Mølck C, et al. Neurochem Res. 2014 Oct;39(10):1862-75. doi: 10.1007/s11064-014-1248-8. Epub 2014 Feb 4. Neurochem Res. 2014. PMID: 24493625

8

Computer-aided discovery of aromatic l-α-amino acids as agonists of the orphan G protein-coupled receptor GPR139.

Isberg V, Andersen KB, Bisig C, Dietz GP, Bräuner-Osborne H, Gloriam DE. Isberg V, et al. J Chem Inf Model. 2014 Jun 23;54(6):1553-7. doi: 10.1021/ci500197a. Epub 2014 May 30. J Chem Inf Model. 2014. PMID: 24826842

9

Functional consequences of glucagon-like peptide-1 receptor cross-talk and trafficking.

Roed SN, Nøhr AC, Wismann P, Iversen H, Bräuner-Osborne H, Knudsen SM, Waldhoer M. Roed SN, et al. J Biol Chem. 2015 Jan 9;290(2):1233-43. doi: 10.1074/jbc.M114.592436. Epub 2014 Dec 1. J Biol Chem. 2015. PMID: 25451942 Free PMC article.

10

Selective Negative Allosteric Modulation Of Metabotropic Glutamate Receptors – A Structural Perspective of Ligands and Mutants.

Harpsøe K, Isberg V, Tehan BG, Weiss D, Arsova A, Marshall FH, Bräuner-Osborne H, Gloriam DE. Harpsøe K, et al. Sci Rep. 2015 Sep 11;5:13869. doi: 10.1038/srep13869. Sci Rep. 2015. PMID: 26359761 Free PMC article.

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