Kolb P - Search Results

1

Comparative Docking to Distinct G Protein-Coupled Receptor Conformations Exclusively Yields Ligands with Agonist Efficacy.

Scharf MM, Bünemann M, Baker JG, Kolb P. Scharf MM, et al. Among authors: kolb p. Mol Pharmacol. 2019 Dec;96(6):851-861. doi: 10.1124/mol.119.117515. Epub 2019 Oct 17. Mol Pharmacol. 2019. PMID: 31624135

2

Limits of ligand selectivity from docking to models: in silico screening for A(1) adenosine receptor antagonists.

Kolb P, Phan K, Gao ZG, Marko AC, Sali A, Jacobson KA. Kolb P, et al. PLoS One. 2012;7(11):e49910. doi: 10.1371/journal.pone.0049910. Epub 2012 Nov 21. PLoS One. 2012. PMID: 23185482 Free PMC article.

3

[Computer-aided design of selective ligands binding to G protein-coupled receptors].

Schmidt D, Kolb P. Schmidt D, et al. Among authors: kolb p. Dtsch Med Wochenschr. 2013 Oct;138(44):2260-4. doi: 10.1055/s-0033-1349483. Epub 2013 Sep 24. Dtsch Med Wochenschr. 2013. PMID: 24065450 Review. German. No abstract available.

4

The mode of agonist binding to a G protein-coupled receptor switches the effect that voltage changes have on signaling.

Rinne A, Mobarec JC, Mahaut-Smith M, Kolb P, Bünemann M. Rinne A, et al. Among authors: kolb p. Sci Signal. 2015 Nov 3;8(401):ra110. doi: 10.1126/scisignal.aac7419. Sci Signal. 2015. PMID: 26535008

5

GPCRdb: the G protein-coupled receptor database - an introduction.

Munk C, Isberg V, Mordalski S, Harpsøe K, Rataj K, Hauser AS, Kolb P, Bojarski AJ, Vriend G, Gloriam DE. Munk C, et al. Among authors: kolb p. Br J Pharmacol. 2016 Jul;173(14):2195-207. doi: 10.1111/bph.13509. Epub 2016 Jun 3. Br J Pharmacol. 2016. PMID: 27155948 Free PMC article. Review.

6

Similarity- and Substructure-Based Development of β₂-Adrenergic Receptor Ligands Based on Unusual Scaffolds.

Schmidt D, Gunera J, Baker JG, Kolb P. Schmidt D, et al. Among authors: kolb p. ACS Med Chem Lett. 2017 Mar 27;8(5):481-485. doi: 10.1021/acsmedchemlett.6b00363. eCollection 2017 May 11. ACS Med Chem Lett. 2017. PMID: 28523097 Free PMC article.

7

The allosteric site regulates the voltage sensitivity of muscarinic receptors.

Hoppe A, Marti-Solano M, Drabek M, Bünemann M, Kolb P, Rinne A. Hoppe A, et al. Among authors: kolb p. Cell Signal. 2018 Jan;42:114-126. doi: 10.1016/j.cellsig.2017.10.011. Epub 2017 Oct 19. Cell Signal. 2018. PMID: 29056499

8

Nanobody-Enabled Reverse Pharmacology on G-Protein-Coupled Receptors.

Pardon E, Betti C, Laeremans T, Chevillard F, Guillemyn K, Kolb P, Ballet S, Steyaert J. Pardon E, et al. Among authors: kolb p. Angew Chem Int Ed Engl. 2018 May 4;57(19):5292-5295. doi: 10.1002/anie.201712581. Epub 2018 Mar 30. Angew Chem Int Ed Engl. 2018. PMID: 29469969

9

Direct targeting of Gα_q and Gα₁₁ oncoproteins in cancer cells.

Annala S, Feng X, Shridhar N, Eryilmaz F, Patt J, Yang J, Pfeil EM, Cervantes-Villagrana RD, Inoue A, Häberlein F, Slodczyk T, Reher R, Kehraus S, Monteleone S, Schrage R, Heycke N, Rick U, Engel S, Pfeifer A, Kolb P, König G, Bünemann M, Tüting T, Vázquez-Prado J, Gutkind JS, Gaffal E, Kostenis E. Annala S, et al. Among authors: kolb p. Sci Signal. 2019 Mar 19;12(573):eaau5948. doi: 10.1126/scisignal.aau5948. Sci Signal. 2019. PMID: 30890659

10

A Taxicab geometry quantification system to evaluate the performance of in silico methods: a case study on adenosine receptors ligands.

Kuder KJ, Michalik I, Kieć-Kononowicz K, Kolb P. Kuder KJ, et al. Among authors: kolb p. J Comput Aided Mol Des. 2020 Jun;34(6):697-707. doi: 10.1007/s10822-020-00301-5. Epub 2020 Feb 28. J Comput Aided Mol Des. 2020. PMID: 32112287 Free PMC article.

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