P450-mediated O-demethylated metabolite is responsible for rat hepatobiliary toxicity of pyridyltriazine-containing PI3K inhibitors.
Subramanian R, Aidasani D, Bailey K, Branstetter D, Everds N, Jiang J, Norman MH, Primack R, Skiles GL, Soto I, Stec MM, Wagner M, Wu T, Zhu X, Lebrec H.
Subramanian R, et al. Among authors: zhu x.
Toxicol Sci. 2014 Nov;142(1):298-310. doi: 10.1093/toxsci/kfu178. Epub 2014 Aug 26.
Toxicol Sci. 2014.
PMID: 25159132