Macrocyclic BACE inhibitors: Optimization of a micromolar hit to nanomolar leads.
Huang Y, Strobel ED, Ho CY, Reynolds CH, Conway KA, Piesvaux JA, Brenneman DE, Yohrling GJ, Moore Arnold H, Rosenthal D, Alexander RS, Tounge BA, Mercken M, Vandermeeren M, Parker MH, Reitz AB, Baxter EW.
Huang Y, et al. Among authors: strobel ed.
Bioorg Med Chem Lett. 2010 May 15;20(10):3158-60. doi: 10.1016/j.bmcl.2010.03.097. Epub 2010 Mar 30.
Bioorg Med Chem Lett. 2010.
PMID: 20399652